SCHEMBL4064085

SCHEMBL4064085

CCN(C=O)C(O)[C@H]1O[C@@H](n2cnc3c(N)nc(N(CCc4ccccc4)C(CCN)CC(N)=O)nc32)[C@H](O)[C@@H]1O

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.42
ADORA1 P30542 4/20 0.42
ADORA2A P29274 4/20 0.42
ADORA2B P29275 3/20 0.42
GNMT Q14749 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3695466 0.82 ADORA3 (0.46) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL3486506 0.81 ADORA2A (0.49) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL8109955 0.79 ADORA2A (0.64) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL2295172 0.79 ADORA2A (0.65) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL258935 0.74 ADORA3 (0.59) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL5964634 0.74 ADORA2A (0.51) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL1976908 0.74 ADORA2A (0.56) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL1081737 0.74 ADORA2A (0.68) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL5964576 0.73 ADORA3 (0.67) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL5689838 0.73 ADORA3 (0.67) ADORA3ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009076580-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT AND PREVENTION OF CARDIOVASCULAR DISEASES THOMAS JEFFERSON UNIVERSITY (US) 2009-06-18 WO disclosed
WO-2008058238-A2 ADENOSINE A1 AND A3 RECEPTOR GENE SEQUENCE VARIATIONS FOR PREDICTING DISEASE OUTCOME AND TREATMENT OUTCOME THOMAS JEFFERSON UNIVERSITY (US) 2008-05-15 WO disclosed