SCHEMBL4065050

SCHEMBL4065050

[CH2]C(O)c1ccc2ncccc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.53
POLB P06746 2/20 0.53
RAB9A P51151 2/20 0.53
ALDH1A1 P00352 7/20 0.50
MAPT P10636 4/20 0.50
HTT P42858 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
CASP1 P29466 2/20 0.50
ATM Q13315 2/20 0.50
KDM4E B2RXH2 2/20 0.50
TP53 P04637 1/20 0.50
HSP90AA1 P07900 1/20 0.50
HSP90AB1 P08238 1/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.50
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MET P08581 3/20 0.44
ALOX15 P16050 1/20 0.44
PLK1 P53350 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31023643 0.85 NPC1 (0.57) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL21709860 0.85 NPC1 (0.57) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL188108 0.82 UGT2B7 (0.56) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL30745165 0.82 UGT2B7 (0.56) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL30063057 0.81 NPC1 (0.49) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL28490619 0.81 NPC1 (0.49) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL13363674 0.81 ALDH1A1 (0.53) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL8917474 0.79 MET (0.54) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL9999689 0.79 MAPT (0.51) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL6852153 0.78 ALDH1A1 (0.52) NPC1POLBRAB9AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1415986-B1 SPIRO ISOBENZOFURANES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS BANYU PHARMA CO LTD (JP) 2009-04-08 EP disclosed
US-7205417-B2 Spiro compounds BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-04-17 US disclosed
CN-1538956-A Spiro compounds ������ҩ��ʽ���� 2004-10-20 CN disclosed