SCHEMBL4065099

SCHEMBL4065099

CNc1cccc(CCOc2ccc(C[C@H](N)C(=O)OC(=O)c3ccc(N4CCCC4)cc3Cl)cc2)n1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.53
ITGAV P06756 19/20 0.53
ITGB1 P05556 18/20 0.53
ITGA5 P08648 18/20 0.53
ITGB6 P18564 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4065095 0.84 ITGB1 (0.76) ITGB3ITGAVITGB1ITGA5
SCHEMBL4065491 0.79 ITGB3 (0.66) ITGB3ITGAVITGB1ITGA5ITGB6
SCHEMBL4254386 0.78 ITGB1 (0.73) ITGB3ITGAVITGB1ITGA5
SCHEMBL14104055 0.77 ITGB3 (0.66) ITGB3ITGAVITGB1ITGA5ITGB6
SCHEMBL4067570 0.77 ITGB3 (0.66) ITGB3ITGAVITGB1ITGA5ITGB6
SCHEMBL4075419 0.76 ITGB3 (0.58) ITGB3ITGAVITGB1ITGA5
Hydrochloric Acid SCHEMBL4193237 0.76 ITGB3 (0.64) ITGB3ITGAVITGB1ITGA5ITGB6
SCHEMBL4739844 0.74 ITGB3 (0.70) ITGB3ITGAVITGB1ITGA5ITGB6
SCHEMBL4398900 0.71 ITGB3 (0.75) ITGB3ITGAVITGB1ITGA5
SCHEMBL4069314 0.70 ITGB3 (0.85) ITGB3ITGAVITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049490-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL]-L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS Astra Zeneca AB (SE) 2009-04-22 EP disclosed
WO-2007141473-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL] -L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS ASTRAZENECA AB (SE) 2007-12-13 WO disclosed