SCHEMBL4065671

SCHEMBL4065671

COC(=O)ON1CCc2c(sc3nc(C)c(C(C)=O)c(-c4ccccc4)c23)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
HPGD P15428 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CACNB4 O00305 1/20 0.40
CACNA1A O00555 1/20 0.40
CACNA1G O43497 1/20 0.40
CACNG3 O60359 1/20 0.40
CACNA1F O60840 1/20 0.40
CACNA1H O95180 1/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
CACNB3 P54284 1/20 0.40
CACNA2D1 P54289 1/20 0.40
CACNG7 P62955 1/20 0.40
CACNA1B Q00975 1/20 0.40
CACNA1D Q01668 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27689851 0.92 KMT2A (0.40) ALDH1A1HPGDKMT2AMEN1CYP3A4
SCHEMBL4067002 0.87 WEE1 (0.44) ALDH1A1HPGDKMT2AMEN1CYP3A4
SCHEMBL27689861 0.83 MAPT (0.42) ALDH1A1HPGDKMT2AMEN1CYP3A4
SCHEMBL27689854 0.80 KMT2A (0.44) KMT2A
SCHEMBL4059322 0.79 P2RX3 (0.52)
SCHEMBL4055917 0.78 KMT2A (0.56) KMT2A
SCHEMBL4059076 0.75 SIGMAR1 (0.43) ALDH1A1HPGDKMT2AMEN1CYP3A4
SCHEMBL4060486 0.71 ALDH1A1 (0.56) ALDH1A1HPGDKMT2AMEN1CYP3A4
SCHEMBL4055022 0.69 ALDH1A1 (0.48) ALDH1A1HPGDKMT2AMEN1CYP3A4
SCHEMBL5505525 0.68 MAPT (0.61) ALDH1A1HPGDKMT2AMEN1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828199-B1 THIENO-PYRIDINE DERIVATIVES AS GABA-B ALLOSTERIC ENHANCERS HOFFMANN LA ROCHE (CH) 2009-05-06 EP claimed