SCHEMBL4065971

SCHEMBL4065971

c1cc(-c2c[nH]nn2)[nH]n1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.46
SCN4A P35499 4/20 0.42
PDPK1 O15530 1/20 0.42
LTA4H P09960 3/20 0.40
POLB P06746 2/20 0.39
PTPN11 Q06124 1/20 0.39
NOTUM Q6P988 3/20 0.38
IDO1 P14902 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
COMT P21964 1/20 0.37
CYP2E1 P05181 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20801657 0.72 NOTUM (0.38) HCAR2SCN4APDPK1LTA4HNOTUM
SCHEMBL87533 0.71
SCHEMBL3068150 0.71 SCN4A (0.62) HCAR2SCN4APDPK1LTA4HPOLB
SCHEMBL132285 0.69
SCHEMBL28099054 0.68 SCN4A (0.43) HCAR2SCN4APDPK1LTA4HPOLB
SCHEMBL949067 0.68
SCHEMBL13078874 0.67 METAP2 (0.32) NPC1RAB9A
SCHEMBL17791787 0.67 HCAR2 (0.61) HCAR2SCN4APDPK1POLBPTPN11
SCHEMBL12075153 0.67 SCN4A (0.52) SCN4APDPK1LTA4HPOLBPTPN11
Bromide SCHEMBL19459238 0.67 LTA4H (0.47) HCAR2SCN4APDPK1LTA4HPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2009184925-A 5-(1H-1,2,3-TRIAZOL-4-YL)-1H-PYRAZOLE DERIVATIVE DAI ICHI SEIYAKU CO LTD 2009-08-20 JP disclosed
WO-2008053602-A1 5-(1H-1,2,3-TRIAZOL-4-YL)-1H-PYRAZOLE DERIVATIVE DAIICHI SANKYO COMPANY, LIMITED (JP) 2008-05-08 WO disclosed