SCHEMBL4066199

SCHEMBL4066199

O=C(O)N1CCC2(CCCCC2)C1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 8/20 0.54
GRM5 P41594 4/20 0.50
SPR P35270 5/20 0.45
USP2 O75604 1/20 0.43
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4073020 0.98 HSD11B1 (0.51) HSD11B1GRM5SPRUSP2CYP3A4
SCHEMBL15618729 0.93 HSD11B1 (0.47) HSD11B1GRM5SPRUSP2CYP3A4
SCHEMBL4072598 0.91 GRM5 (0.59) HSD11B1GRM5SPRUSP2CYP3A4
Hydrochloric Acid SCHEMBL30751767 0.91 HSD11B1 (0.46) HSD11B1GRM5SPRUSP2CYP3A4
SCHEMBL18422376 0.89 GRM5 (0.49) HSD11B1GRM5USP2CYP3A4CYP2C19
SCHEMBL22032412 0.89 GRM5 (0.56) HSD11B1GRM5SPRUSP2CYP3A4
SCHEMBL29418104 0.89 HSD11B1 (0.42) HSD11B1GRM5SPRUSP2CYP3A4
SCHEMBL4062010 0.86 HSD11B1 (0.45) HSD11B1GRM5SPRUSP2CYP3A4
SCHEMBL30329203 0.84 GRM5 (0.52) HSD11B1GRM5SPRUSP2CYP3A4
SCHEMBL4066092 0.84 GRM5 (0.52) HSD11B1GRM5SPRUSP2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12599672-B2 KRAS proteolysis targeting chimeras PAQ Therapeutics Inc. (US) 2026-04-14 US disclosed
US-20260062443-A1 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS ALEXION PHARMA INC (US) 2026-03-05 US disclosed
WO-2025224085-A1 COMPOUNDS CAPABLE OF ACTING ON S1R AS WELL AS ON SEH AND USES THEREOF UNIVERSITAT DE BARCELONA (ES) 2025-10-30 WO disclosed
US-20250144225-A1 KRAS Proteolysis Targeting Chimeras PAQ Therapeutics Inc. (US) 2025-05-08 US disclosed
US-20230212152-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. 2023-07-06 US disclosed
EP-4161902-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2023-04-12 EP disclosed
CN-111601807-B Exo-azaspiro inhibitors of MENIN-MLL interactions 詹森药业有限公司 2023-03-31 CN disclosed
US-11524940-B1 Inhibitors of cysteine proteases and methods of use thereof Pardes Biosciences, Inc. (US) 2022-12-13 US disclosed
US-11396517-B1 Exo-aza spiro inhibitors of menin-MLL interaction JANSSEN PHARMACEUTICA NV (BE) 2022-07-26 US disclosed
EP-2520568-A1 Spirocyclic nitriles as inhibitors of protease SANOFI (FR) 2012-11-07 EP disclosed
EP-2032535-B1 SPIROCYCLIC NITRILES AS PROTEASE INHIBITORS SANOFI SA (FR) 2012-08-01 EP disclosed
EP-2032535-A1 SPIROCYCLIC NITRILES AS PROTEASE INHIBITORS Sanofi-Aventis (FR) 2009-03-11 EP disclosed
WO-2007137738-A1 SPIROCYCLIC NITRILES AS PROTEASE INHIBITORS SANOFI-AVENTIS (DE) 2007-12-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12599672-B2 KRAS proteolysis targeting chimeras KRAS, HRAS, NRAS HSD11B1 3145/4885GRM5 4554/4885SPR 3999/4885
US-20260062443-A1 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS C9, SSB, C1S HSD11B1 2670/4885GRM5 1304/4885SPR 3098/4885
US-20250144225-A1 KRAS Proteolysis Targeting Chimeras KRAS, HRAS, NRAS HSD11B1 3197/4885GRM5 4186/4885SPR 1900/4885
US-11396517-B1 Exo-aza spiro inhibitors of menin-MLL interaction BMI1, MLLT1, EED HSD11B1 2531/4885GRM5 2427/4885SPR 1818/4885
US-11524940-B1 Inhibitors of cysteine proteases and methods of use thereof CTRL, CTSV, CTSL HSD11B1 3036/4885GRM5 4411/4885SPR 1005/4885
US-20230212152-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF CTRL, CTSL, CTSV HSD11B1 2299/4885GRM5 4524/4885SPR 1830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.