SCHEMBL4068537

SCHEMBL4068537

COc1ccc2nccc(N3CC[N]CC3)c2n1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP8B1 Q9UNU6 1/20 0.41
NCF1 P14598 2/20 0.40
ACVR1 Q04771 1/20 0.38
KCNH2 Q12809 3/20 0.36
EHMT2 Q96KQ7 2/20 0.36
EHMT1 Q9H9B1 2/20 0.36
GAA P10253 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1222623 0.85 NCF1 (0.57) CYP8B1NCF1
SCHEMBL1222834 0.83 CYP2C19 (0.46) CYP8B1NCF1ACVR1KCNH2
SCHEMBL1223241 0.81 CHRNB2 (0.53) CYP8B1NCF1
SCHEMBL4068487 0.80 EHMT2 (0.41) CYP8B1KCNH2EHMT2EHMT1
SCHEMBL4069340 0.80 KCNH2 (0.42) KCNH2EHMT2EHMT1
SCHEMBL1224035 0.80 CYP2C19 (0.43) CYP8B1NCF1ACVR1KCNH2
SCHEMBL1222688 0.78 CYP2C19 (0.54) CYP8B1ACVR1KCNH2
SCHEMBL3634872 0.78 CYP2C19 (0.54) CYP8B1ACVR1KCNH2
SCHEMBL3636416 0.78 CYP2C19 (0.54) CYP8B1ACVR1KCNH2
SCHEMBL3168429 0.78 CYP8B1 (0.50) CYP8B1ACVR1KCNH2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1605938-B1 Antibacterial derivatives of napthydrin and quinoline GLAXO GROUP LTD (GB) 2009-02-11 EP claimed
EP-1605938-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2006-11-22 EP claimed
EP-1605938-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2005-12-21 EP claimed
WO-2004087145-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2004-10-14 WO claimed