SCHEMBL4068635

SCHEMBL4068635

COc1cc(OC)c(C(C)C)cc1-c1ccccc1NS(=O)(=O)Cc1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 3/20 0.46
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPK1 P28482 1/20 0.45
PTK2B Q14289 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CYP17A1 P05093 2/20 0.44
MCL1 Q07820 1/20 0.42
LPAR1 Q92633 2/20 0.40
BRD4 O60885 1/20 0.40
NPC1 O15118 2/20 0.39
TSHR P16473 1/20 0.38
PARP14 Q460N5 1/20 0.38
MRGPRX1 Q96LB2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13848473 0.91 ALDH1A1 (0.54) ALDH1A1KDM4EMAPK1PTK2BHPGD
SCHEMBL13848410 0.87 CYP17A1 (0.46) PTGES2ALDH1A1KDM4EMAPK1PTK2B
SCHEMBL4544247 0.84 HSD17B10 (0.47) ALDH1A1MAPK1PTK2BHPGDHSD17B10
SCHEMBL13848251 0.83 PTGES2 (0.53) PTGES2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL13848077 0.82 CYP17A1 (0.49) PTGES2ALDH1A1KDM4EMAPK1PTK2B
SCHEMBL13848277 0.81 PARP14 (0.46) PTGES2HPGDHSD17B10CYP17A1PARP14
SCHEMBL13848266 0.80 L3MBTL1 (0.54) ALDH1A1KDM4EMAPK1HPGDCYP17A1
SCHEMBL13848445 0.75 MRGPRX1 (0.43) CYP17A1LPAR1MRGPRX1
SCHEMBL13848365 0.74 ALDH1A1 (0.61) ALDH1A1HSD17B10
SCHEMBL4544124 0.74 CYP17A1 (0.48) ALDH1A1MAPK1PTK2BHPGDCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009066060-A2 4-SUBSTITUTED-6-ISOPROPYL-BENZENE-1,3-DIOL COMPOUNDS AND THEIR USE TOPOTARGET A/S (DK) 2009-05-28 WO disclosed
WO-2009066060-A2 4-SUBSTITUTED-6-ISOPROPYL-BENZENE-1,3-DIOL COMPOUNDS AND THEIR USE TOPOTARGET A/S (DK) 2009-05-28 WO disclosed