Fluticasone

Fluticasone

SCHEMBL4069

C[C@@H]1C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)SCF

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 14/20 1.00
PGR P06401 5/20 0.76
AR P10275 5/20 0.76
CYP3A4 P08684 4/20 0.76
HIF1A Q16665 3/20 0.76
SMN1; SMN2 Q16637 2/20 0.76
ABCB11 O95342 1/20 0.76
ALDH1A1 P00352 1/20 0.76
MAPT P10636 1/20 0.76
RAB9A P51151 1/20 0.76
MEN1 O00255 1/20 0.75
ALOX15 P16050 1/20 0.75
KMT2A Q03164 1/20 0.75
NR3C2 P08235 2/20 0.73
NR1I2 O75469 1/20 0.73
ADORA3 P0DMS8 1/20 0.73
CNR1 P21554 1/20 0.66
PTGS1 P23219 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluticasone SCHEMBL65401 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4HIF1A
Fluticasone SCHEMBL14135286 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4HIF1A
Fluticasone SCHEMBL2231799 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4HIF1A
Fluticasone SCHEMBL28888601 0.99 NR3C1 (0.98) NR3C1PGRARCYP3A4HIF1A
Fluticasone SCHEMBL28821706 0.99 NR3C1 (0.98) NR3C1PGRARCYP3A4HIF1A
Fluticasone SCHEMBL28935320 0.98 NR3C1 (0.97) NR3C1PGRARCYP3A4HIF1A
Fluticasone SCHEMBL27674669 0.97 NR3C1 (0.95) NR3C1PGRARCYP3A4HIF1A
Fluticasone SCHEMBL896670 0.97 NR3C1 (0.93) NR3C1PGRARCYP3A4HIF1A
Fluticasone SCHEMBL29113054 0.96 NR3C1 (0.92) NR3C1PGRARCYP3A4HIF1A
Fluticasone SCHEMBL3365958 0.95 NR3C1 (0.91) NR3C1PGRARCYP3A4HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 40234 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423298-B1 None US claimed
EP-4747263-A1 LIPID NANOPARTICLES AND USES THEREOF University of Connecticut (US) 2026-05-27 EP claimed
US-20260137656-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
US-20260137657-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
US-20260130899-A1 METHOD OF TREATMENT FOR PREVENTION OF GLUCOCORTICOID TOXICITY AND/OR ENHANCEMENT OF MUSCLE REGENERATION VIA NEUTROPHIL ELASTASE INHIBITION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2026-05-14 US claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
US-20260125686-A1 COMPOSITIONS AND METHODS FOR MODULATION OF CFTR CYSTIC FIBROSIS FOUND (US) 2026-05-07 US claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-0577760-A1 SEQUENTIAL DOSING OF ANTIFUNGAL AND ANTIINFLAMMATORY COMPOSITIONS GLAXO WELLCOME INC. (US) 1994-01-12 EP claimed
EP-0278174-B1 USE OF FLUTICASONE PROPIONATE IN THE PREPARATION OF A PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF BOWEL DISEASES GLAXO GROUP LIMITED (GB) 1993-03-10 EP claimed
US-5174475-A Dispensing a first component followed by second without adjustment GLAXO INC. (US) 1992-12-29 US claimed
WO-1992018133-A1 METHOD OF TREATMENT USING STEROID MOUTHWASH EISEN DRORE (US) 1992-10-29 WO claimed
WO-1992017183-A1 SEQUENTIAL DOSING OF ANTIFUNGAL AND ANTIINFLAMMATORY COMPOSITIONS GLAXO INC. (US) 1992-10-15 WO claimed
EP-0470154-A1 DRY POWDER INHALATION DEVICE. RIKER LABORATORIES INC (US) 1992-02-12 EP claimed
US-5049389-A Non-phospholipd lipid, delivery by inhalation LIPOSOME TECHNOLOGY, INC. (US) 1991-09-17 US claimed
WO-1990013328-A1 DRY POWDER INHALATION DEVICE RIKER LABORATORIES, INC. (US) 1990-11-15 WO claimed
WO-1990013327-A1 DRY POWDER INHALATION DEVICE RIKER LABORATORIES, INC. (US) 1990-11-15 WO claimed
WO-1990006775-A1 A NOVEL NONPHOSPHOLIPID LIPOSOME COMPOSITION FOR SUSTAINED RELEASE OF DRUGS LIPOSOME TECHNOLOGY, INC. (US) 1990-06-28 WO claimed