SCHEMBL4069491

SCHEMBL4069491

CC(=O)c1cc(-n2cc3c(n2)CCN(CC(=O)N2CCN(C4CCC4)CC2)C3)ccn1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HRH3 Q9Y5N1 5/20 0.36
SLC6A9 P48067 1/20 0.34
PARP1 P09874 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ENPP2 Q13822 1/20 0.33
F10 P00742 1/20 0.33
KDM4E B2RXH2 2/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
ALDH1A1 P00352 1/20 0.33
IRAK4 Q9NWZ3 2/20 0.32
ACHE P22303 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748854 0.90 SLC6A9 (0.43) HTTNPSR1HRH3SLC6A9PARP1
SCHEMBL4067642 0.88 SLC6A9 (0.43) HTTNPSR1HRH3SLC6A9PARP1
SCHEMBL4061339 0.88 HRH3 (0.37) HTTNPSR1HRH3SLC6A9PARP1
SCHEMBL13748862 0.88 HTT (0.35) HTTNPSR1HRH3SLC6A9PARP1
SCHEMBL13749068 0.88 CYP2C9 (0.38) HTTNPSR1HRH3SLC6A9PARP1
SCHEMBL13748931 0.87 PDK2 (0.36) HTTNPSR1HRH3SLC6A9PARP1
SCHEMBL13749350 0.86 SLC6A9 (0.39) HTTNPSR1HRH3SLC6A9PARP1
SCHEMBL13748292 0.86 HRH3 (0.43) HTTNPSR1HRH3PARP1SMN1; SMN2
SCHEMBL1017656 0.85 HTT (0.39) HTTNPSR1HRH3PARP1SMN1; SMN2
SCHEMBL4069495 0.85 SMO (0.40) HRH3SMN1; SMN2ENPP2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100120-A2 PYRIDINYL-SUBSTITUTED PIPERAZINYL OXOETHYL TETRAHYDROPYRAZOLOPYRIDINES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed