SCHEMBL13749068

SCHEMBL13749068

COc1cc(-n2cc3c(n2)CCN(CC(=O)N2CCN(C4CCC4)CC2)C3)ccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.38
NR1H2 P55055 2/20 0.38
NR1H3 Q13133 2/20 0.38
CYP2D6 P10635 2/20 0.38
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
SLC6A9 P48067 1/20 0.36
HRH3 Q9Y5N1 4/20 0.35
ACVR1 Q04771 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
OPRM1 P35372 1/20 0.35
CACNA2D1 P54289 1/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HTT P42858 1/20 0.35
KDM4E B2RXH2 1/20 0.34
PARP1 P09874 1/20 0.34
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748854 0.89 SLC6A9 (0.43) ALDH1A1KMT2ASLC6A9HRH3CHRM4
SCHEMBL4069491 0.88 HTT (0.39) ALDH1A1TSHRKMT2ASLC6A9HRH3
SCHEMBL4061339 0.87 HRH3 (0.37) ALDH1A1SLC6A9HRH3NPSR1HTT
SCHEMBL4067642 0.87 SLC6A9 (0.43) ALDH1A1KMT2ASLC6A9HRH3NPSR1
SCHEMBL13748862 0.87 HTT (0.35) ALDH1A1SLC6A9HRH3NPSR1HTT
SCHEMBL13748931 0.86 PDK2 (0.36) ALDH1A1KMT2ASLC6A9HRH3NPSR1
SCHEMBL1016129 0.85 ALDH1A1 (0.47) ALDH1A1TSHRKMT2AHRH3KDM4E
SCHEMBL13749350 0.85 SLC6A9 (0.39) SLC6A9HRH3CHRM1CHRM4NPSR1
SCHEMBL13748292 0.85 HRH3 (0.43) ALDH1A1KMT2AHRH3NPSR1HTT
SCHEMBL1071102 0.85 HRH3 (0.37) ALDH1A1TSHRKMT2AHRH3NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100120-A2 PYRIDINYL-SUBSTITUTED PIPERAZINYL OXOETHYL TETRAHYDROPYRAZOLOPYRIDINES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed