SCHEMBL4072093

SCHEMBL4072093

COc1cc(C=NN(CC(=O)CN(N=Cc2cc(OC)cc(OC)c2)C(=O)O)C(=O)O)cc(OC)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
G6PC1 P35575 2/20 0.41
CYP1B1 Q16678 3/20 0.38
CYP1A1 P04798 2/20 0.38
BACE1 P56817 1/20 0.37
PTGS2 P35354 2/20 0.36
NQO2 P16083 2/20 0.35
FFAR1 O14842 1/20 0.35
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
ABL1 P00519 2/20 0.34
BCR P11274 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4079893 0.71 G6PC1 (0.45) G6PC1CYP1B1PTGS2ABL1BCR
SCHEMBL10706017 0.65 CHRM5 (0.63) CYP1B1CYP1A1PTGS2NQO2ABL1
SCHEMBL13569071 0.64 CYP1A2 (0.53) MEN1NPC1MAPTRAB9AKMT2A
SCHEMBL22925041 0.63 CYP1B1 (0.52) CYP1B1CYP1A1PTGS2NQO2ABL1
SCHEMBL13569101 0.63 POLB (0.57) BACE1KDM4EMEN1GAAMAPT
SCHEMBL5383597 0.63 CYP1B1 (0.47) CYP1B1CYP1A1PTGS2NQO2ABL1
SCHEMBL5383595 0.63 CYP1B1 (0.47) CYP1B1CYP1A1PTGS2NQO2ABL1
SCHEMBL21386596 0.62 CYP1B1 (0.56) CYP1B1CYP1A1PTGS2NQO2ABCG2
SCHEMBL13128174 0.62 CYP1B1 (0.56) CYP1B1CYP1A1PTGS2NQO2ABL1
SCHEMBL6251820 0.62 CYP1A1 (0.50) CYP1B1CYP1A1PTGS2NQO2ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009155362-A1 SMALL MOLECULE HEMATOPOIETIC GROWTH FACTOR MIMETIC COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2009-12-23 WO disclosed