SCHEMBL4072134

SCHEMBL4072134

C[C@H](Nc1nc(N)c(F)c(-c2cc(C3CC3)n[nH]2)n1)c1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 12/20 0.48
JAK2 O60674 1/20 0.41
JAK3 P52333 1/20 0.41
GRK6 P43250 6/20 0.39
ADRA1D P25100 1/20 0.39
HTR2C P28335 1/20 0.39
HTR7 P34969 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
HTR6 P50406 1/20 0.39
AURKA O14965 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4071743 0.91 NTRK1 (0.47) NTRK1JAK2JAK3GRK6ADRA1D
SCHEMBL4074269 0.85 NTRK1 (0.49) NTRK1JAK2JAK3GRK6ADRA1D
SCHEMBL4152477 0.84 NTRK1 (0.55) NTRK1JAK2JAK3
SCHEMBL30010123 0.83 NTRK1 (0.52) NTRK1JAK2JAK3
SCHEMBL23217059 0.83 NTRK1 (0.52) NTRK1JAK2JAK3
SCHEMBL4067495 0.81 IGF1R (0.43) NTRK1HTR7
SCHEMBL4075051 0.80 MAPK13 (0.41) NTRK1
SCHEMBL2511149 0.79 NTRK1 (0.41) NTRK1JAK2JAK3GRK6ADRA1D
SCHEMBL4491060 0.79 NTRK1 (0.41) NTRK1JAK2JAK3GRK6ADRA1D
SCHEMBL3341173 0.78 NTRK1 (0.55) NTRK1JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1686999-B1 PYRAZOLE DERIVATIVES AS INHIBITORS OF RECEPTOR TYROSINE KINASES ASTRAZENECA AB (SE) 2009-07-01 EP disclosed