SCHEMBL4072555

SCHEMBL4072555

COCCc1c(C#N)cnc2ccccc12.Cc1c(C#N)cnc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.43
MAP2K1 Q02750 4/20 0.39
RAF1 P04049 2/20 0.39
EGFR P00533 4/20 0.36
ERBB2 P04626 3/20 0.36
LDHA P00338 1/20 0.36
SRC P12931 5/20 0.35
ABL1 P00519 1/20 0.35
FLT1 P17948 1/20 0.35
KDR P35968 1/20 0.35
SYK P43405 1/20 0.35
MYC P01106 1/20 0.35
NSD2 O96028 3/20 0.34
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4063577 0.94 LRRK2 (0.48) LRRK2MAP2K1RAF1EGFRERBB2
SCHEMBL3151307 0.82 LRRK2 (0.58) LRRK2MAP2K1RAF1EGFRERBB2
SCHEMBL4246880 0.78 LRRK2 (0.38) LRRK2MAP2K1RAF1EGFRERBB2
SCHEMBL27668508 0.76 TLR7 (0.47) LRRK2MAP2K1RAF1TSHR
SCHEMBL4572184 0.75 LRRK2 (0.54) LRRK2MAP2K1RAF1SRC
SCHEMBL3156282 0.72 LRRK2 (0.50) LRRK2MAP2K1RAF1EGFRERBB2
SCHEMBL4231806 0.72 LRRK2 (0.50) LRRK2MAP2K1RAF1SRC
SCHEMBL27668262 0.72 LRRK2 (0.57) LRRK2MAP2K1RAF1EGFRERBB2
SCHEMBL20178365 0.69 LRRK2 (0.54) LRRK2MAP2K1RAF1EGFRERBB2
SCHEMBL20494995 0.69 ALDH1A1 (0.43) LDHAMYCTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1706412-A4 NOVEL PYRIDINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME SK CHEMICALS CO LTD (KR) 2009-03-18 EP disclosed
EP-1706412-A1 NOVEL PYRIDINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME SK Chemicals, Co., Ltd. (KR) 2006-10-04 EP disclosed
WO-2005063768-A1 NOVEL PYRIDINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME SK CHEMICALS, CO., LTD. (KR) 2005-07-14 WO disclosed