SCHEMBL4246880

SCHEMBL4246880

COCCc1c(C#N)cnc2ccccc12.O=C1OCCc2c1cnc1ccccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.38
DPP4 P27487 2/20 0.33
KCNH2 Q12809 2/20 0.33
MYC P01106 1/20 0.33
EED O75530 7/20 0.33
SUZ12 Q15022 7/20 0.33
EZH2 Q15910 7/20 0.33
RBBP4 Q09028 6/20 0.33
AEBP2 Q6ZN18 6/20 0.33
SLC2A1 P11166 1/20 0.33
MAP2K1 Q02750 2/20 0.32
RAF1 P04049 1/20 0.32
EGFR P00533 3/20 0.32
ABL1 P00519 1/20 0.32
SRC P12931 1/20 0.32
FLT1 P17948 1/20 0.32
KDR P35968 1/20 0.32
SYK P43405 1/20 0.32
POLB P06746 1/20 0.32
ERBB2 P04626 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4063577 0.83 LRRK2 (0.48) LRRK2MYCMAP2K1RAF1EGFR
SCHEMBL4072632 0.78 ALDH1A1 (0.42) LRRK2ALDH1A1CYP1A2
SCHEMBL4072555 0.78 LRRK2 (0.43) LRRK2MYCMAP2K1RAF1EGFR
SCHEMBL4572184 0.67 LRRK2 (0.54) LRRK2DPP4KCNH2MAP2K1RAF1
SCHEMBL27668508 0.65 TLR7 (0.47) LRRK2MAP2K1RAF1ALDH1A1CYP1A2
SCHEMBL7412699 0.65 ALOX5 (0.42)
SCHEMBL4231806 0.64 LRRK2 (0.50) LRRK2MAP2K1RAF1SRCPOLB
SCHEMBL3156282 0.64 LRRK2 (0.50) LRRK2DPP4KCNH2MAP2K1RAF1
SCHEMBL27668262 0.63 LRRK2 (0.57) LRRK2DPP4KCNH2MAP2K1RAF1
SCHEMBL20494995 0.63 ALDH1A1 (0.43) MYCALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1706412-A4 NOVEL PYRIDINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME SK CHEMICALS CO LTD (KR) 2009-03-18 EP disclosed
EP-1706412-A1 NOVEL PYRIDINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME SK Chemicals, Co., Ltd. (KR) 2006-10-04 EP disclosed
WO-2005063768-A1 NOVEL PYRIDINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME SK CHEMICALS, CO., LTD. (KR) 2005-07-14 WO disclosed