SCHEMBL4072947

SCHEMBL4072947

FC(F)Oc1cccc(N2C[CH]CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
RECQL P46063 1/20 0.40
RXRA P19793 6/20 0.40
GRIN1 Q05586 6/20 0.40
GRIN2B Q13224 6/20 0.40
GALR2 O43603 1/20 0.38
GALR1 P47211 1/20 0.38
DRD1 P21728 1/20 0.37
NOTUM Q6P988 1/20 0.36
ADRB1 P08588 1/20 0.36
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
KDM2B Q8NHM5 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4067558 0.91 GALR2 (0.42) KDM4ERECQLRXRAGRIN1GRIN2B
SCHEMBL4064747 0.90 KDM4E (0.42) KDM4ERECQLRXRAGRIN1GRIN2B
SCHEMBL4064662 0.82 ALDH1A1 (0.45) RXRAGRIN1GRIN2BGALR2DRD1
SCHEMBL4067230 0.79 ADRB1 (0.58) KDM4EADRB1KMT2ANPC1MAPT
SCHEMBL17893764 0.76 KDM4E (0.44) KDM4ERECQLRXRAGRIN1GRIN2B
SCHEMBL5761993 0.76 ADRB1 (0.64) ADRB1MAPT
Hydrochloric Acid SCHEMBL6501617 0.75 ADRB1 (0.62) ADRB1MAPT
Hydrochloric Acid SCHEMBL6414607 0.75 ADRB1 (0.62) ADRB1MAPT
SCHEMBL4072922 0.75 BPTF (0.50) NOTUMKMT2AMAPT
SCHEMBL4067061 0.73 ALDH1A1 (0.42) KDM4ERXRAGRIN1GRIN2BGALR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1415986-B1 SPIRO ISOBENZOFURANES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS BANYU PHARMA CO LTD (JP) 2009-04-08 EP disclosed
US-7205417-B2 Spiro compounds BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-04-17 US disclosed