SCHEMBL4073305

SCHEMBL4073305

CC(C)(C(=O)Nc1nc2ccccc2s1)S(=O)(=O)c1ccc(Cl)cc1F.CC(C)(C(=O)Nc1nsc(-c2ccccc2)n1)S(=O)(=O)c1ccc(Cl)cc1F.CC(C)(C)c1nnc(NC(=O)C(C)(C)S(=O)(=O)c2ccc(Cl)cc2F)s1.CCc1ccnc(NC(=O)C(C)(C)S(=O)(=O)c2ccc(Cl)cc2F)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
LCK P06239 1/20 0.35
PIK3CA P42336 3/20 0.34
AKT1 P31749 2/20 0.34
MTOR P42345 1/20 0.34
PIK3C3 Q8NEB9 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
CNR2 P34972 2/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CNR1 P21554 1/20 0.33
DHODH Q02127 1/20 0.33
CSNK1D P48730 2/20 0.33
RAB9A P51151 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4070531 0.87 CNR2 (0.38) MAPTALDH1A1KDM4EHPGDPIK3C3
SCHEMBL4069812 0.85 MEN1 (0.41) ALDH1A1PIK3C3MEN1KMT2ACNR2
SCHEMBL1464075 0.78 NPC1 (0.47) MAPTALDH1A1KDM4EHPGDMEN1
SCHEMBL1465943 0.75 DHODH (0.55) MAPTKDM4EMEN1KMT2ACNR2
SCHEMBL1464745 0.75 PKM (0.43) PIK3C3CNR2CNR1MAPK14
SCHEMBL1465181 0.74 MEN1 (0.53) MAPTALDH1A1CYP2C9CYP2C19MEN1
SCHEMBL3960775 0.70 CNR2 (0.42) MAPTALDH1A1HPGDCNR2CNR1
SCHEMBL1465579 0.69 ALDH1A1 (0.50) MAPTALDH1A1HPGDCNR2GRM4
SCHEMBL1466234 0.66 MEN1 (0.52) MAPTALDH1A1KDM4ECYP2C9HPGD
SCHEMBL1465871 0.66 CNR2 (0.53) MAPTALDH1A1KDM4EHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081905-A2 SULFONYL COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR Boehringer Ingelheim International GmbH (DE) 2009-07-29 EP claimed
WO-2008014199-A2 SULFONYL COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-01-31 WO claimed