Cefazolin

Cefazolin

SCHEMBL40736

Cc1nnc(SCC2=C(C(=O)O)N3C(=O)[C@@H](NC(=O)Cn4cnnn4)[C@H]3SC2)s1.[NaH]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Cefazolin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.98
PTGS2 P35354 1/20 0.98
SLC22A6 Q4U2R8 1/20 0.98
SLC22A8 Q8TCC7 1/20 0.98
SLC22A11 Q9NSA0 1/20 0.98
MAPT P10636 9/20 0.84
TDP1 Q9NUW8 9/20 0.84
ABCC4 O15439 1/20 0.84
BLM P54132 1/20 0.84
CYP3A4 P08684 1/20 0.84
NFKB1 P19838 1/20 0.84
HSD17B10 Q99714 1/20 0.84
PTGS1 P23219 1/20 0.72
PDE4A P27815 1/20 0.72
KDR P35968 1/20 0.72
POLB P06746 9/20 0.70
ALDH1A1 P00352 4/20 0.68
MAPK1 P28482 1/20 0.68
KMT2A Q03164 3/20 0.68
MEN1 O00255 2/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cefazolin SCHEMBL6364010 1.00 LMNA (0.98) LMNAPTGS2SLC22A6SLC22A8SLC22A11
Cefazolin SCHEMBL28254869 1.00 LMNA (0.98) LMNAPTGS2SLC22A6SLC22A8SLC22A11
Cefazolin SCHEMBL1698164 0.99 LMNA (0.97) LMNAPTGS2SLC22A6SLC22A8SLC22A11
Cefazolin SCHEMBL2911037 0.99 LMNA (0.97) LMNAPTGS2SLC22A6SLC22A8SLC22A11
Cefazolin SCHEMBL11031717 0.99 LMNA (1.00) LMNAPTGS2SLC22A6SLC22A8SLC22A11
Cefazolin SCHEMBL16072809 0.99 LMNA (1.00) LMNAPTGS2SLC22A6SLC22A8SLC22A11
Cefazolin SCHEMBL4930576 0.99 LMNA (1.00) LMNAPTGS2SLC22A6SLC22A8SLC22A11
Cefazolin SCHEMBL3894722 0.99 LMNA (1.00) LMNAPTGS2SLC22A6SLC22A8SLC22A11
Cefazolin SCHEMBL2842 0.99 LMNA (1.00) LMNAPTGS2SLC22A6SLC22A8SLC22A11
Cefazolin SCHEMBL3424683 0.99 LMNA (1.00) LMNAPTGS2SLC22A6SLC22A8SLC22A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5950 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122036754-A Cefazolin sodium method for preparing anhydrous substance 河北合佳创新医药科技有限公司 2026-05-15 CN claimed
WO-2025111413-A1 TREATMENT FOR SKIN DISORDERS Mycotechnology, Inc. (US) 2025-05-30 WO claimed
CN-115015212-B Spectral detection method for antiviral and antibacterial drug residues in water 广东省科学院测试分析研究所(中国广州分析测试中心) 2025-05-23 CN claimed
CN-119970732-A Antibacterial composition with synergistic effect and application thereof 南京工业大学 2025-05-13 CN claimed
US-12274830-B2 Nitric oxide inhalation therapy for infants with bronchiolitis BEYOND AIR LTD (IL) 2025-04-15 US claimed
CN-119780320-A Method for measuring acetyl hydrazine in cefazolin sodium by high performance liquid chromatography-tandem mass spectrometry 新发药业有限公司 2025-04-08 CN claimed
CN-119757629-A Method for detecting related substances in cefazolin sodium 武汉九州钰民医药科技有限公司 2025-04-04 CN claimed
CN-119733055-A Composition of beta-lactam inhibitor and cephalosporin medicine, and preparation method and application thereof 福建泽瑞药业有限公司 2025-04-01 CN claimed
CN-119643765-A Analysis method of cefazolin sodium and cefazolin sodium polymer impurities for injection 上海上药新亚药业有限公司 2025-03-18 CN claimed
CN-119510634-A Polymer analysis method of cefazolin sodium for injection 哈药集团技术中心 2025-02-25 CN claimed
EP-0327081-A2 Alpha-crystals of cefazolin sodium FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-08-09 EP claimed
CN-87106855-A The manufacture method of composition for oral liquid 1988-04-20 CN claimed
CN-86105639-A The preparation method of rectally dosage form 1987-02-25 CN claimed
US-4486411-A SYNERGISTIC MIXTURES WITH BETA-LACTAM ANTIBIOTICS PFIZER INC. (US) 1984-12-04 US claimed
US-4146971-A Method of preparing a rapidly dissolving powder of sterile crystalline cefazolin sodium for parenteral administration ELI LILLY AND COMPANY (US) 1979-04-03 US claimed
US-4104391-A Method of preparing stable sterile ampoules of crystalline cephalosporins for parenteral administration ELI LILLY AND COMPANY (US) 1978-08-01 US claimed
US-4104470-A Crystallization process for cefazolin sodium ELI LILLY AND COMPANY (US) 1978-08-01 US claimed
US-4029655-A Method of preparing stable sterile crystalline cephalosporins for parenteral administration ELI LILLY AND COMPANY (US) 1977-06-14 US claimed
US-4002748-A Method of preparing sterile essentially amorphous cefazolin for reconstitution for parenteral administration ELI LILLY AND COMPANY (US) 1977-01-11 US claimed
US-3937655-A Method for preparing stable β-lactam-type-antibiotic susceptibility test discs ELI LILLY AND COMPANY (US) 1976-02-10 US claimed