SCHEMBL4076309

SCHEMBL4076309

CC(CC(=O)N(C)c1cccnc1)C(=O)NC1CCC(Cc2ccc(Cl)cc2)(N(C)C)CC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 2/20 0.39
PYGL P06737 1/20 0.38
AVPR1A P37288 4/20 0.36
TRPV1 Q8NER1 1/20 0.36
CYP3A4 P08684 2/20 0.35
TSHR P16473 2/20 0.35
SLC1A3 P43003 1/20 0.35
SLC1A2 P43004 1/20 0.35
SLC1A1 P43005 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
NOTUM Q6P988 1/20 0.34
OXTR P30559 1/20 0.34
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206292 0.74 KMT2A (0.42) C3AR1PYGLMEN1KMT2AKDM4E
SCHEMBL2984799 0.72 TDP1 (0.44) AVPR1AOXTR
SCHEMBL2976914 0.72 TSHR (0.49) AVPR1ATSHR
SCHEMBL2991416 0.70 AVPR1A (0.41) AVPR1AOXTR
SCHEMBL4861833 0.69 MEN1 (0.46) CYP3A4TSHRMEN1KMT2A
SCHEMBL206987 0.68 POLB (0.56) CYP3A4TSHRMEN1KMT2A
SCHEMBL207560 0.68 POLB (0.41) AVPR1AMEN1KMT2A
SCHEMBL2979024 0.68 LMNA (0.49) AVPR1ATSHRMEN1KMT2A
SCHEMBL4079453 0.67 LMNA (0.43) AVPR1ATSHROXTR
SCHEMBL205911 0.66 ALDH1A1 (0.40) TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed