SCHEMBL4077193

SCHEMBL4077193

COc1ccc(-c2ccccc2OC(N)=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.51
HDAC4 P56524 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
FGFR1 P11362 1/20 0.51
SRC P12931 1/20 0.51
FGFR2 P21802 1/20 0.51
FGFR4 P22455 1/20 0.51
FGFR3 P22607 1/20 0.51
ABL1 P00519 1/20 0.49
ABCB1 P08183 1/20 0.49
BCR P11274 1/20 0.49
TUBB4A P04350 1/20 0.48
TUBB P07437 1/20 0.48
TUBA3C P0DPH7 1/20 0.48
TUBA1B P68363 1/20 0.48
TUBA4A P68366 1/20 0.48
TUBB4B P68371 1/20 0.48
TUBB3 Q13509 1/20 0.48
TUBB2A Q13885 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8065693 0.87 BACE1 (0.54) BACE1HDAC4HDAC2HDAC8FGFR1
SCHEMBL1717103 0.85 BACE1 (0.71) BACE1HDAC4HDAC2HDAC8ABL1
SCHEMBL8065696 0.85 BACE1 (0.53) BACE1HDAC4HDAC2HDAC8FGFR1
SCHEMBL7647143 0.83 LMNA (0.50) SYKRAB9ASMN1; SMN2MAPTLMNA
SCHEMBL274364 0.83 FABP3 (0.53) RAB9ASMN1; SMN2TP53LMNAMAPK1
SCHEMBL31448682 0.83 FABP3 (0.49) RAB9ASMN1; SMN2TP53LMNAMAPK1
SCHEMBL27469798 0.81 NCOA1 (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL20573270 0.81 SLC6A4 (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL27615667 0.81 CYP1A2 (0.49) HDAC4HDAC2HDAC8ABCB1NPC1
SCHEMBL20573256 0.81 BACE1 (0.52) BACE1HDAC4HDAC2HDAC8SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3029026-B1 NOVEL BIPHENYL DERIVATIVE AND METHOD FOR PREPARING SAME DONG A ST CO LTD (KR) 2018-12-05 EP claimed
EP-3029026-A1 NOVEL BIPHENYL DERIVATIVE AND METHOD FOR PREPARING SAME Dong-A ST Co., Ltd. (KR) 2016-06-08 EP disclosed
EP-1711183-A4 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LTD (GB) 2009-04-01 EP disclosed
EP-1711183-A2 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2006-10-18 EP disclosed
WO-2005067537-A2 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2005-07-28 WO disclosed
CN-1638761-A Azetidine derivatives as CCR-3 receptor antagonists NOVARTIS AG (CH) 2005-07-13 CN disclosed