SCHEMBL4077534

SCHEMBL4077534

NC(=O)c1ccc(C(=O)N(c2cccc(Nc3nccc(-c4cccnc4)n3)c2)c2ccccc2N)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 17/20 0.64
PDGFRB P09619 6/20 0.64
HDAC1 Q13547 2/20 0.64
HDAC3 O15379 1/20 0.64
KDR P35968 1/20 0.64
HDAC4 P56524 1/20 0.64
HDAC7 Q8WUI4 1/20 0.64
HDAC2 Q92769 1/20 0.64
HDAC10 Q969S8 1/20 0.64
HDAC11 Q96DB2 1/20 0.64
HDAC8 Q9BY41 1/20 0.64
HDAC6 Q9UBN7 1/20 0.64
HDAC9 Q9UKV0 1/20 0.64
HDAC5 Q9UQL6 1/20 0.64
MAPK8 P45983 2/20 0.57
PIK3CG P48736 1/20 0.57
GSK3B P49841 1/20 0.57
CAMKK2 Q96RR4 1/20 0.57
BCR P11274 14/20 0.55
ABL2 P42684 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4087392 0.87 PDGFRB (0.54) ABL1PDGFRBHDAC1HDAC3KDR
SCHEMBL4086274 0.87 PDGFRB (0.67) ABL1PDGFRBHDAC1HDAC3KDR
SCHEMBL4080340 0.79 PDGFRA (0.56) ABL1PDGFRBHDAC1HDAC3KDR
SCHEMBL4895454 0.78 ABL1 (0.80) ABL1PDGFRBMAPK8PIK3CGGSK3B
SCHEMBL4087658 0.78 ABL1 (1.00) ABL1PDGFRBHDAC1HDAC3KDR
Hydrochloric Acid SCHEMBL27711429 0.77 ABL1 (0.79) ABL1PDGFRBMAPK8PIK3CGGSK3B
SCHEMBL4903328 0.77 MAPK8 (0.81) ABL1PDGFRBHDAC1MAPK8PIK3CG
Hydrochloric Acid SCHEMBL27708725 0.77 ABL1 (0.77) ABL1PDGFRBMAPK8PIK3CGGSK3B
SCHEMBL4086310 0.73 HDAC1 (0.84) ABL1PDGFRBHDAC1HDAC3KDR
SCHEMBL2944431 0.72 CAMKK2 (0.77) ABL1MAPK8PIK3CGGSK3BCAMKK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2060565-A1 Novel bifunctional compounds which inhibit protein kinases and histone deacetylases 4SC AG (DE) 2009-05-20 EP disclosed