SCHEMBL4078446

SCHEMBL4078446

Oc1cc(-c2ccccc2)cc(Cl)c1C(O)C1CCN(c2ncccn2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
TSHR P16473 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SLC6A7 Q99884 4/20 0.40
KDM4E B2RXH2 3/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTR1A P08908 1/20 0.39
MAPT P10636 2/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
MALT1 Q9UDY8 1/20 0.38
SLC6A3 Q01959 2/20 0.37
LMNA P02545 1/20 0.37
DPP4 P27487 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3812208 0.83 ALDH1A1 (0.44) ALDH1A1TSHRMEN1KMT2ASLC6A7
SCHEMBL3832885 0.80 HTR1A (0.41) ALDH1A1TSHRMEN1KMT2ASLC6A7
SCHEMBL3585163 0.76 SLC6A7 (0.56) SLC6A7SLC6A3
SCHEMBL4488282 0.76 SLC6A7 (0.56) SLC6A7SLC6A3
SCHEMBL4074249 0.76 SLC6A7 (0.56) SLC6A7SLC6A3
SCHEMBL4234609 0.76 SLC6A7 (0.50) SLC6A7MALT1SLC6A3DPP4DPP8
SCHEMBL4075764 0.76 ESR2 (0.36) ALDH1A1TSHRMEN1KMT2ASLC6A7
SCHEMBL4234602 0.76 SLC6A7 (0.50) SLC6A7MALT1SLC6A3DPP4DPP8
SCHEMBL4497275 0.76 SLC6A7 (0.50) SLC6A7MALT1SLC6A3DPP4DPP8
SCHEMBL4075757 0.76 ESR2 (0.36) ALDH1A1TSHRMEN1KMT2ASLC6A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2084145-A2 (S)-PHENYL(HETEROCYCLE)METHANOL-BASED COMPOUNDS, COMPOSITIONS COMPRISING THEM AND METHODS OF THEIR USE Lexicon Pharmaceuticals, Inc. (US) 2009-08-05 EP disclosed
WO-2008067120-A2 (S)-PHENYL(HETEROCYCLE)METHANOL-BASED COMPOUNDS, COMPOSITIONS COMPRISING THEM AND METHODS OF THEIR USE LEXICON PHARMACEUTICALS, INC. (US) 2008-06-05 WO disclosed