SCHEMBL4079403

SCHEMBL4079403

CCCCCCNC(=O)N1CC(OC(c2ccc(Cl)cc2)c2ccc(Cl)cc2)C1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.47
FAAH O00519 5/20 0.46
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
EPHX1 P07099 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5818620 0.86 FAAH (0.50) FAAHCNR1CNR2
SCHEMBL4075740 0.84 KMT2A (0.45) NAMPTCNR1CNR2
SCHEMBL4084791 0.82 FAAH (0.47) FAAHCNR1CNR2
SCHEMBL4635589 0.81 FAAH (0.48) FAAHCNR1CNR2
SCHEMBL4635584 0.81 FAAH (0.48) FAAHCNR1CNR2
SCHEMBL4084892 0.80 FAAH (0.52) FAAHCNR1CNR2EPHX1
SCHEMBL4078545 0.79 NAAA (0.43) NAMPTFAAHCNR1CNR2
SCHEMBL4078364 0.79 CNR1 (0.55) FAAHCNR1
SCHEMBL4079362 0.78 GAA (0.48) FAAHCNR1CNR2
SCHEMBL4636071 0.78 FAAH (0.43) FAAHCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620395-B1 AZETIDINECARBOXAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CB1 RECEPTOR MEDIATED DISORDERS VERNALIS RES LTD (GB) 2009-12-30 EP disclosed
US-7504522-B2 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disorders VERNALIS RESEARCH LIMITED (GB) 2009-03-17 US disclosed
US-20070054891-A1 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disorders VERNALIS RESEARCH LIMAITED (GB) 2007-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070054891-A1 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disorders CNR1, CNR2, GPR119 NAMPT 3230/4885FAAH 8/4885CNR1 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.