SCHEMBL4079865

SCHEMBL4079865

O=C(O)N1CCNc2ncc(Br)cc2C1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABHD6 Q9BV23 1/20 0.38
NNMT P40261 2/20 0.38
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PIK3C3 Q8NEB9 1/20 0.33
AHR P35869 1/20 0.32
BRS3 P32247 4/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
GRM5 P41594 1/20 0.31
OPRK1 P41145 1/20 0.30
ALDH1A1 P00352 2/20 0.30
GAA P10253 2/20 0.30
MAPK1 P28482 1/20 0.30
MAPT P10636 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
GPR142 Q7Z601 1/20 0.30
FNTA P49354 2/20 0.30
FNTB P49356 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL724954 0.81 MAPK1 (0.54) ABHD6MAPK1MAPTFNTAFNTB
SCHEMBL14995412 0.78 ABHD6 (0.38) ABHD6HPGDHTTALDH1A1
SCHEMBL13320471 0.77 BRD4 (0.33) NNMTPIK3C3GRM5
SCHEMBL723952 0.75 ABHD6 (0.49) ABHD6HPGDHTTSMN1; SMN2GRM5
Bromide SCHEMBL2844387 0.75 BRD4 (0.32) NNMTGRM5
SCHEMBL725593 0.75 IDH1 (0.40) BRS3L3MBTL1MAPK1
SCHEMBL2844900 0.74 MAPK1 (0.46) ABHD6HPGDMAPK1MAPTFNTA
SCHEMBL2843141 0.74 ESR1 (0.36) NNMTHPGDALDH1A1FNTAFNTB
SCHEMBL2843054 0.74 HTR3E (0.39) SMN1; SMN2GRM5MAPT
SCHEMBL21591731 0.73 ABHD6 (0.59) ABHD6HPGDHTTSMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054422-A1 ACRYLAMIDE DERIVATIVES AS FAB I INHIBITORS Affinium Pharmaceuticals, Inc. (CA) 2009-05-06 EP disclosed
WO-2008009122-A1 ACRYLAMIDE DERIVATIVES AS FAB I INHIBITORS AFFINIUM PHARMACEUTICALS, INC. (CA) 2008-01-24 WO disclosed