SCHEMBL4083873

SCHEMBL4083873

CCCC1=C(C(=O)OCC)C(c2ccc(CC)s2)NC(=O)N1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 4/20 0.62
ADORA2A P29274 1/20 0.62
MAPK1 P28482 1/20 0.57
HSD17B10 Q99714 1/20 0.57
PKM P14618 1/20 0.49
CASP1 P29466 1/20 0.48
POLB P06746 2/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
TP53 P04637 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
KDM4E B2RXH2 1/20 0.44
APEX1 P27695 1/20 0.44
ESR2 Q92731 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4253445 0.87 ADORA2B (0.59) ADORA2BADORA2AMAPK1HSD17B10PKM
SCHEMBL4263419 0.86 PKM (0.65) ADORA2BMAPK1HSD17B10PKMCASP1
SCHEMBL3005564 0.81 PKM (0.75) ADORA2BADORA2AMAPK1HSD17B10PKM
SCHEMBL10113271 0.79 HSD17B10 (0.74) ADORA2BADORA2AMAPK1HSD17B10POLB
SCHEMBL2999682 0.79 ADORA2B (0.69) ADORA2BADORA2AMAPK1HSD17B10CASP1
SCHEMBL2994443 0.76 ADORA2B (0.75) ADORA2BADORA2AMAPK1HSD17B10
SCHEMBL10113267 0.76 HSD17B10 (0.72) ADORA2BADORA2AMAPK1HSD17B10POLB
SCHEMBL10113258 0.74 TSHR (0.75) ADORA2BADORA2AMAPK1HSD17B10POLB
SCHEMBL10113282 0.73 MAPK1 (0.76) ADORA2BADORA2AMAPK1HSD17B10POLB
SCHEMBL2999627 0.72 MAPT (0.65) HSD17B10CASP1POLBALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed