SCHEMBL4084095

SCHEMBL4084095

O=C(O)CCCC(=O)N1CCN(Cc2coc3ccccc23)CC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.52
DRD2 P14416 8/20 0.50
DRD4 P21917 8/20 0.50
DRD3 P35462 8/20 0.50
ALDH1A1 P00352 5/20 0.45
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 2/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
HTR1A P08908 2/20 0.44
GPR6 P46095 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
APP P05067 1/20 0.43
TSHR P16473 1/20 0.43
HTR7 P34969 1/20 0.43
LMNA P02545 2/20 0.42
HTT P42858 1/20 0.42
MAPT P10636 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4075730 0.74 HTR2B (0.60) DRD2DRD4DRD3HTR1A
SCHEMBL5763082 0.74 MAOB (0.50) KDM4ESMN1; SMN2
SCHEMBL1750627 0.74 SIGMAR1 (0.58) SIGMAR1DRD2DRD4DRD3ALDH1A1
SCHEMBL1387431 0.73 ALDH1A1 (0.62) SIGMAR1DRD2DRD4DRD3ALDH1A1
SCHEMBL13772456 0.73 SIGMAR1 (0.58) SIGMAR1DRD2DRD4DRD3ALDH1A1
SCHEMBL28262836 0.71 ALDH1A1 (0.57) SIGMAR1DRD2DRD4DRD3ALDH1A1
SCHEMBL5762073 0.71 MAOB (0.53) KDM4E
SCHEMBL4074069 0.70 MEN1 (0.60) ALDH1A1KDM4EHTR1ASMN1; SMN2TSHR
SCHEMBL4072689 0.69 ALDH1A1 (0.70) ALDH1A1KDM4EHSD17B10TSHRHTR7
SCHEMBL7295692 0.69 SIGMAR1 (1.00) SIGMAR1ALDH1A1HSD17B10HTR1ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed