SCHEMBL4087295

SCHEMBL4087295

N#Cc1cccc(CCc2cc(N)[nH]n2)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.43
NOS1 P29475 3/20 0.42
HRH3 Q9Y5N1 1/20 0.42
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
KCNJ1 P48048 1/20 0.38
KCNH2 Q12809 1/20 0.38
LRRK2 Q5S007 1/20 0.38
GLA P06280 1/20 0.38
NOS2 P35228 2/20 0.37
ADRA2C P18825 1/20 0.37
VNN1 O95497 1/20 0.36
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL64650 0.78 BACE1 (0.49) MPONOS1KCNH2ALDH1A1
SCHEMBL2154019 0.78 GLA (0.53) NOS1HRH3CYP19A1CYP11B1CYP11B2
SCHEMBL3939288 0.77 MPO (0.46) MPONOS1HRH3CYP19A1CYP11B1
SCHEMBL63824 0.74 TAAR1 (0.54)
SCHEMBL4010143 0.73 FOLH1 (0.46) CYP4F2CYP4A11
SCHEMBL9878817 0.72 HRH3 (0.46) MPONOS1HRH3CYP19A1CYP11B1
SCHEMBL6950852 0.72 TSHR (0.52) HRH3CYP19A1CYP11B1CYP11B2KCNJ1
SCHEMBL63191 0.72 CYP2A6 (0.51) MPOHRH3NOS2
SCHEMBL6420561 0.72 ADRA2C (0.47) NOS1HRH3CYP19A1CYP11B1CYP11B2
SCHEMBL3939419 0.71 CYP4F2 (0.54) MPOCYP4F2CYP4A11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009056886-A1 PYRIMIDINE DERIVATIVES AND THEIR USE AS MODULATORS OF FGFR ACTIVITY ASTRAZENECA AB (SE) 2009-05-07 WO disclosed