SCHEMBL6950852

SCHEMBL6950852

N#Cc1cccc(CCc2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
FFAR1 O14842 2/20 0.51
FFAR4 Q5NUL3 1/20 0.51
MAOA P21397 4/20 0.50
MAOB P27338 4/20 0.50
ALDH1A1 P00352 1/20 0.49
KDM1A O60341 1/20 0.49
LMNA P02545 1/20 0.49
GLA P06280 1/20 0.49
KCNJ1 P48048 1/20 0.48
KCNH2 Q12809 1/20 0.48
DRD2 P14416 2/20 0.47
DRD3 P35462 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
CYP19A1 P11511 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2154019 0.94 GLA (0.53) TSHRFFAR1FFAR4MAOAMAOB
SCHEMBL6962952 0.92 DRD2 (0.49) TSHRFFAR1FFAR4MAOAMAOB
SCHEMBL6951637 0.90 FAAH (0.50) TSHRFFAR1FFAR4MAOAMAOB
SCHEMBL6960752 0.90 FAAH (0.50) TSHRFFAR1FFAR4MAOAMAOB
SCHEMBL9900679 0.86 ALDH1A1 (0.48) FFAR1FFAR4MAOAMAOBALDH1A1
SCHEMBL28248372 0.85 HTR2B (0.54) FFAR1FFAR4MAOAMAOBALDH1A1
SCHEMBL28865565 0.85 HTR2B (0.50) FFAR1FFAR4MAOAMAOBALDH1A1
SCHEMBL7450600 0.84 CLK4 (0.50) MAOBALDH1A1GLAMEN1KMT2A
SCHEMBL24358855 0.83 HTR2B (0.49) TSHRFFAR1FFAR4GLAKCNJ1
SCHEMBL29732423 0.83 HTR2B (0.49) TSHRFFAR1FFAR4GLAKCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10449174-B2 Aryl isonitrile compounds as a new class of potent, broad-spectrum antifungal compounds PURDUE RESEARCH FOUNDATION (US) 2019-10-22 US disclosed
US-20170181997-A1 ARYL ISONITRILE COMPOUNDS AS A NEW CLASS OF POTENT, BROAD-SPECTRUM ANTIFUNGAL COMPOUNDS PURDUE RESEARCH FOUNDATION (US) 2017-06-29 US disclosed
CN-106190930-A One strain lactobacillus delbruockii subspecies bulgaricus MGA17 6 and application thereof 内蒙古农业大学 2016-12-07 CN disclosed
CN-102726455-A Botanical nematocide and preparation method thereof DAQING COLLEGE HEILONGJIANG ACADEMY OF SCIENCE 2012-10-17 CN disclosed
EP-0711762-B1 PROCESS FOR PRODUCING TETRAZOLE COMPOUNDS SUMITOMO CHEMICAL CO (JP) 2003-08-06 EP disclosed
US-6277998-B1 REACTING 2-CYANO-4-OXO-4H-BENZOPYRAN COMPOUND WITH HYDROGEN SULFIDE AND THEN REACTING PROUDCT WITH ALKYL HALIDE; REACTING THE PRODUCT WITH HYDRAZINE OR ITS SALT AND THEN WITH NITROUS ACID COMPOUND TO OBTAIN TETRAZOLE COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2001-08-21 US disclosed
US-6191289-B1 REACTING A 4-OXO-4H-BENZOPYRAN GROUP SUBSTITUTED WITH AMIDE OR A PHENYL GROUP IN ITS 2 POSITION IS REACTED WITH ANHYDROUS HYDRAZINE OR SALT IN PRESENCE OF CATALYST FOLLOWED BY REACTING WITH NITROUS ACID OR SALT TO FORM TETRAZOLE COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2001-02-20 US disclosed
US-5874593-A SULFUR CONTAINING AMIDE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-02-23 US disclosed
EP-0711762-A1 PROCESS FOR PRODUCING TETRAZOLE COMPOUND AND INTERMEDIATE THEREFOR SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-05-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10449174-B2 Aryl isonitrile compounds as a new class of potent, broad-spectrum antifungal compounds AHR, CYP3A4, NAT1 TSHR 3640/4885FFAR1 2450/4885FFAR4 1177/4885
US-20170181997-A1 ARYL ISONITRILE COMPOUNDS AS A NEW CLASS OF POTENT, BROAD-SPECTRUM ANTIFUNGAL COMPOUNDS AHR, CYP3A4, NAT1 TSHR 3640/4885FFAR1 2450/4885FFAR4 1177/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.