Formamide

Formamide

SCHEMBL4091594

Cc1ccnc(C)c1C.NC=O

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 6/20 0.50
NOS3 P29474 5/20 0.50
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CCR8 P51685 1/20 0.37
CYP2A6 P11509 1/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
P2RX7 Q99572 1/20 0.32
NOS1 P29475 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
LIMK1 P53667 1/20 0.31
SIRT3 Q9NTG7 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ALDH1A1 P00352 1/20 0.30
NR2F2 P24468 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7488 0.86
Iodide SCHEMBL27713885 0.84 NOS2 (0.54) NOS2NOS3CCR1CCR5CCR8
Hydrochloric Acid SCHEMBL27389327 0.84 NOS2 (0.54) NOS2NOS3CCR1CCR5CCR8
Hydrochloric Acid SCHEMBL1936574 0.84 NOS2 (0.54) NOS2NOS3CCR1CCR5CCR8
Fluoride SCHEMBL2020932 0.84 NOS2 (0.54) NOS2NOS3CCR1CCR5CCR8
Bromide SCHEMBL10623434 0.84 NOS2 (0.54) NOS2NOS3CCR1CCR5CCR8
Iodide SCHEMBL11070568 0.84 NOS2 (0.54) NOS2NOS3CCR1CCR5CCR8
SCHEMBL29125217 0.84
Ammonia Solution, Strong SCHEMBL22612697 0.84 NOS2 (0.54) NOS2NOS3CCR1CCR5CCR8
SCHEMBL10993290 0.83 CYP2A6 (0.46) NOS2NOS3CCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867636-A1 PYRIDYLMETHYLSULFONE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2007-12-19 EP claimed
EP-1867636-B1 PYRIDYLMETHYLSULFONE DERIVATIVE DAIICHI SANKYO CO LTD (JP) 2013-06-05 EP disclosed
US-20090149439-A1 PYRIDYLMETHYSULFONE DERIVATIVE DAIICHI SANKYO COMPANY LIMITED (JP) 2009-06-11 US disclosed
EP-1867636-A1 PYRIDYLMETHYLSULFONE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2007-12-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090149439-A1 PYRIDYLMETHYSULFONE DERIVATIVE APP, IAPP, BACE1 NOS2 938/4885NOS3 1038/4885CCR1 4830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.