SCHEMBL4092525

SCHEMBL4092525

CC(c1ncc[nH]1)N(C)C

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
FPR2 P25090 4/20 0.36
NISCH Q9Y2I1 2/20 0.35
F2RL1 P55085 4/20 0.35
TXN P10599 1/20 0.34
TXNRD1 Q16881 1/20 0.34
TAAR1 Q96RJ0 2/20 0.34
MTOR P42345 1/20 0.33
ADK P55263 1/20 0.33
MMP1 P03956 1/20 0.33
MMP3 P08254 1/20 0.33
MMP7 P09237 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL369263 0.84 ADRA2A (0.41) ADRA2AADRA2BADRA2CALDH1A1SMN1; SMN2
SCHEMBL12233238 0.80 F2RL1 (0.38) ADRA2AADRA2BADRA2CALDH1A1SMN1; SMN2
SCHEMBL6039544 0.79 ADRA2A (0.38) ADRA2AADRA2BADRA2CALDH1A1SMN1; SMN2
SCHEMBL6039548 0.79 ADRA2A (0.40) ADRA2AADRA2BADRA2CALDH1A1SMN1; SMN2
SCHEMBL29046781 0.77 ADRA2A (0.53) ADRA2AADRA2BADRA2CALDH1A1SMN1; SMN2
SCHEMBL189942 0.77
SCHEMBL10225887 0.76 TAAR1 (0.48) ADRA2AADRA2BADRA2CSMN1; SMN2TXN
Hydrochloric Acid SCHEMBL10681958 0.75 ADRA2A (0.47) ADRA2AADRA2BADRA2CALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL4259010 0.75 ADRA2A (0.47) ADRA2AADRA2BADRA2CALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL27564991 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8461167-B2 Acetylenic heteroaryl compounds ARIAD PHARMACEUTICALS, INC. (US) 2013-06-11 US disclosed
US-20090176781-A1 Acetylenic Heteroaryl Compounds ARIAD PHARMACEUTICALS, INC. 2009-07-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176781-A1 Acetylenic Heteroaryl Compounds NAT1, AADAC, ACACA ADRA2A 808/4885ADRA2B 648/4885ADRA2C 423/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.