SCHEMBL409430

SCHEMBL409430

Cc1cccc(-c2nn3ccccc3c2-c2ccnc3cc(C(=O)NCCN4CCOCC4)ccc23)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 6/20 0.49
HPGDS O60760 3/20 0.46
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
PTGER4 P35408 2/20 0.44
TGFBR2 P37173 3/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
POLB P06746 1/20 0.43
GAK O14976 1/20 0.43
RIPK2 O43353 1/20 0.43
MAP4K4 O95819 1/20 0.43
KDR P35968 1/20 0.43
ACVR1B P36896 1/20 0.43
CSNK1A1 P48729 1/20 0.43
CSNK1D P48730 1/20 0.43
CSNK1E P49674 1/20 0.43
TGFB2 P61812 1/20 0.43
MAPK14 Q16539 1/20 0.43
MINK1 Q8N4C8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL409683 0.96 TGFBR1 (0.48) TGFBR1HPGDSTGFBR2L3MBTL1GAK
SCHEMBL414211 0.90 TGFBR1 (0.53) TGFBR1TGFBR2GAKRIPK2MAP4K4
SCHEMBL412977 0.89 TGFBR1 (0.51) TGFBR1TGFBR2GAKRIPK2MAP4K4
SCHEMBL414681 0.88 TGFBR1 (0.51) TGFBR1TGFBR2POLBGAKRIPK2
SCHEMBL413710 0.86 TGFBR1 (0.49) TGFBR1TGFBR2L3MBTL1POLBGAK
SCHEMBL412319 0.86 TGFBR1 (0.61) TGFBR1PTGER4TGFBR2GAKRIPK2
SCHEMBL412491 0.85 TGFBR1 (0.57) TGFBR1TGFBR2GAKRIPK2MAP4K4
SCHEMBL413597 0.84 TGFBR1 (0.48) TGFBR1TGFBR2GAKRIPK2MAP4K4
SCHEMBL412989 0.84 TGFBR1 (0.47) TGFBR1TGFBR2GAKRIPK2MAP4K4
SCHEMBL412295 0.83 NAMPT (0.50) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120021519-A1 EFFICIENT INDUCTION OF PLURIPOTENT STEM CELLS USING SMALL MOLECULE COMPOUNDS PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-26 US disclosed