SCHEMBL4095688

SCHEMBL4095688

COc1ccc(Cn2c(=O)c(OC)nn(-c3cccc(N(C(C)=O)c4ccccc4)c3)c2=O)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
TSHR P16473 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ROCK2 O75116 1/20 0.36
TP53 P04637 1/20 0.35
CMA1 P23946 3/20 0.35
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
CTSK P43235 1/20 0.34
P2RX7 Q99572 1/20 0.34
NPBWR1 P48145 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580890 0.83 LMNA (0.42) ALDH1A1TSHRMEN1KMT2A
SCHEMBL3592958 0.78 MAPK14 (0.45) ALDH1A1TSHRSMN1; SMN2HPGDMEN1
SCHEMBL3581370 0.77 PDE10A (0.37) ROCK2CMA1CTSKNPBWR1
SCHEMBL3589496 0.76 MAPT (0.43) MEN1KMT2AROCK2TP53NPBWR1
SCHEMBL3577324 0.75 SMN1; SMN2 (0.42) ALDH1A1SMN1; SMN2ROCK2POLBL3MBTL1
SCHEMBL3577788 0.72 ROCK2 (0.45) ROCK2P2RX7
SCHEMBL3590298 0.72 MAPK1 (0.49) TP53P2RX7
SCHEMBL3588015 0.72 PKM (0.42) ALDH1A1TSHRKMT2AROCK2POLB
SCHEMBL3580070 0.70 GPBAR1 (0.40) TSHRHSD17B10POLBCTSKNPBWR1
SCHEMBL3588105 0.70 ROCK2 (0.41) MEN1KMT2AROCK2TP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2104670-A2 NOVEL TRIAZINEDIONE DERIVATIVES AS GABA-B RECEPTOR MODULATORS Addex Pharma SA (CH) 2009-09-30 EP disclosed
WO-2008056257-A2 NOVEL TRIAZINEDIONE DERIVATIVES AS GABA-B RECEPTOR MODULATORS ADDEX PHARMA S.A (CH) 2008-05-15 WO disclosed