SCHEMBL4099395

SCHEMBL4099395

CC(c1c(Br)c2ccccc2c[n+]1O)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.40
LMNA P02545 3/20 0.40
TP53 P04637 2/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 4/20 0.34
HTT P42858 3/20 0.34
POLB P06746 2/20 0.33
GAA P10253 2/20 0.33
KMT2A Q03164 2/20 0.33
NPC1 O15118 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
DNMT1 P26358 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2729617 0.85 TDP1 (0.38) TDP1LMNATP53MAPK1NPSR1
SCHEMBL4091324 0.76 NCEH1 (0.38) POLBNPC1
SCHEMBL2729350 0.72 ALDH1A1 (0.33) TDP1LMNATP53MAPK1NPSR1
SCHEMBL2730524 0.71 NPSR1 (0.39) TDP1LMNATP53MAPK1NPSR1
SCHEMBL6923510 0.67 POLB (0.49) TDP1LMNAALDH1A1POLBGAA
SCHEMBL6923507 0.67 POLB (0.49) TDP1LMNAALDH1A1POLBGAA
SCHEMBL31706143 0.64 LMNA (0.47) TDP1LMNATP53MAPK1NPSR1
SCHEMBL2002901 0.64 LMNA (0.47) TDP1LMNATP53MAPK1NPSR1
SCHEMBL2002904 0.64 LMNA (0.47) TDP1LMNATP53MAPK1NPSR1
SCHEMBL14729729 0.64 LMNA (0.47) TDP1LMNATP53MAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061696-A1 5 -CYANO-4, 6 -DIAMINOPYRIMIDINE OR 6 -AMINOPURINE DERIVATIVES AS PI3K- DELTA INHIBITORS AMGEN INC. (US) 2012-05-10 WO disclosed