SCHEMBL411156

SCHEMBL411156

CC(=O)c1cccc(C(=O)O)c1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
ALOX15 P16050 1/20 0.50
KDM4E B2RXH2 4/20 0.47
HPGD P15428 4/20 0.47
HSD17B10 Q99714 3/20 0.47
CA12 O43570 5/20 0.45
CA1 P00915 5/20 0.45
CA2 P00918 5/20 0.45
CA7 P43166 5/20 0.45
CA9 Q16790 5/20 0.45
CA4 P22748 3/20 0.45
AKR1C3 P42330 1/20 0.45
CA14 Q9ULX7 3/20 0.44
MAPK1 P28482 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
KMT2A Q03164 1/20 0.44
TSHR P16473 2/20 0.44
HMGB1 P09429 2/20 0.44
NAPRT Q6XQN6 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8879116 0.98 ALDH1A1 (0.48) ALDH1A1ALOX15KDM4EHPGDHSD17B10
SCHEMBL598165 0.95 CA12 (0.48) ALDH1A1ALOX15KDM4EHPGDHSD17B10
SCHEMBL2953498 0.91 ALDH1A1 (0.50) ALDH1A1ALOX15KDM4EHPGDHSD17B10
Acetic Acid SCHEMBL27417814 0.91 ALDH1A1 (0.55) ALDH1A1ALOX15KDM4EHPGDHSD17B10
SCHEMBL23288 0.88 ALDH1A1 (0.63) ALDH1A1ALOX15KDM4EHPGDHSD17B10
SCHEMBL711798 0.88 ALDH1A1 (0.63) ALDH1A1ALOX15KDM4EHPGDHSD17B10
SCHEMBL15049648 0.86 ALDH1A1 (0.55) ALDH1A1ALOX15KDM4EHPGDHSD17B10
SCHEMBL723062 0.85 ALDH1A1 (0.60) ALDH1A1ALOX15KDM4EHPGDHSD17B10
SCHEMBL1535448 0.85 ALDH1A1 (0.60) ALDH1A1ALOX15KDM4EHPGDHSD17B10
Hydrochloric Acid SCHEMBL3459326 0.85 ALDH1A1 (0.60) ALDH1A1ALOX15KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1315 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240150794-A1 Methods for Delivering a Cargo Into a Cell Trince bv (BE) 2024-05-09 US claimed
CN-117979941-A Liquid filled capsule with two-phase liquid fill 龙沙格林伍德有限公司 2024-05-03 CN claimed
EP-4340801-A1 LIQUID FILLED CAPSULE WITH TWO PHASE LIQUID FILL Lonza Greenwood LLC (US) 2024-03-27 EP claimed
EP-4305183-A1 METHODS FOR DELIVERING A CARGO INTO A CELL Trince bv (BE) 2024-01-17 EP claimed
CN-117396611-A Method for delivering a cargo into a cell 成思有限责任公司 2024-01-12 CN claimed
WO-2023214018-A1 GASTRO-RETENTIVE SWELLABLE SUSTAINED RELEASE COMPOSITION GALENIX INNOVATIONS (FR) 2023-11-09 WO claimed
WO-2023187176-A1 METHOD FOR DELIVERING A CARGO INTO CELL Trince bv (BE) 2023-10-05 WO claimed
US-20230225979-A1 SOLID ORAL COMPOSITIONS COMPRISING COMPOSITE MONOLITHIC MATRICES FOR CHRONOTROPIC ADMINISTRATION OF ACTIVE INGREDIENTS IN THE GASTROINTESTINAL TRACT MOGON PHARMACEUTICALS SAGL (CH) 2023-07-20 US claimed
EP-4149438-A1 SOLID ORAL COMPOSITIONS COMPRISING COMPOSITE MONOLITHIC MATRICES FOR CHRONOTROPIC ADMINISTRATION OF ACTIVE INGREDIENTS IN THE GASTROINTESTINAL TRACT Mogon Pharmaceuticals Sagl (CH) 2023-03-22 EP claimed
EP-4132473-A1 PHARMACEUTICAL COMPOSITION FOR TREATING INFLAMMATORY BOWEL DISEASES Cvasthera (FR) 2023-02-15 EP claimed
US-4832958-A HYPOTENSIVE AGENTS PHARLYSE SOCIETE ANONYME (LU) 1989-05-23 US claimed
US-4786506-A MULTISTEP COATING AND GRANULATION PROCESS ISTITUTO GENTILI S.P.A. (IT) 1988-11-22 US claimed
US-4766012-A DISSOLVING COATING BY SALT FORMATION, DISPERSION OF DRUG PARTICLES, ACIDIFICATION TO PRECIPITATE COATING FARMACEUTICI FORMENTI S.P.A. (IT) 1988-08-23 US claimed
EP-0212751-A2 Process for the microencapsulation of a medicament, medicament so prepared and pharmaceutical compositions comprising it FARMACEUTICI FORMENTI S.p.A. (IT) 1987-03-04 EP claimed
EP-0063132-B1 NEW GALENICAL ADMINISTRATION FORM OF METOCLOPRAMIDE, METHOD FOR ITS PREPARATION AND MEDICAMENT COMPRISING THIS NEW FORM LARUELLE, Claude (FR) 1986-07-30 EP claimed
US-4490407-A SPRAYING, DRYING, TO FORM COATED GRANULES LABORATOIRE L. LAFON (FR) 1984-12-25 US claimed
US-4432966-A SUSTAINED RELEASE ROUSSEL-UCLAF (FR) 1984-02-21 US claimed
EP-0094123-A2 Therapeutic granules THE PROCTER & GAMBLE COMPANY (US) 1983-11-16 EP claimed
EP-0092060-A1 Pharmaceutical products in sustained-release form, and their preparation process LABORATORI PROPHIN Industria Chimica Farmaceutica S.p.A. (IT) 1983-10-26 EP claimed
EP-0030172-B1 PROCESS FOR PREPARING RHESUS ANTIGEN, MEDICINE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE ANTIGEN AND ADMINISTRATION FORMS OEUVRE REGIONALE DE TRANSFUSION SANGUINE DE TOULOUSE (FR) 1983-02-09 EP claimed