SCHEMBL411279

SCHEMBL411279

OC(Cn1c2ccccc2c2ccccc21)Cn1c2ccc(Br)cc2c2cc(Br)ccc21

nearest known ligand 0.78

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.78
MEN1 O00255 1/20 0.78
RAD52 P43351 1/20 0.78
BACE1 P56817 2/20 0.71
DNM1 Q05193 9/20 0.66
MAPT P10636 3/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
BAX Q07812 1/20 0.62
TP53 P04637 1/20 0.60
CYP3A4 P08684 1/20 0.60
ALOX15 P16050 1/20 0.60
MAPK1 P28482 1/20 0.60
P2RX3 P56373 1/20 0.59
HTT P42858 2/20 0.56
NPSR1 Q6W5P4 2/20 0.56
LMNA P02545 1/20 0.56
POLB P06746 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16923672 0.93 KMT2A (0.69) KMT2AMEN1RAD52BACE1DNM1
SCHEMBL16923735 0.92 KMT2A (0.68) KMT2AMEN1RAD52BACE1DNM1
SCHEMBL410834 0.92 DNM1 (0.73) KMT2AMEN1RAD52BACE1DNM1
SCHEMBL6815606 0.92 MEN1 (0.88) KMT2AMEN1RAD52BACE1DNM1
SCHEMBL608294 0.86 BAX (0.88) KMT2AMEN1RAD52BACE1DNM1
SCHEMBL1305296 0.86 MEN1 (0.78) KMT2AMEN1RAD52BACE1DNM1
SCHEMBL607333 0.86 BAX (0.88) KMT2AMEN1RAD52BACE1DNM1
SCHEMBL607334 0.86 BAX (0.88) KMT2AMEN1RAD52BACE1DNM1
SCHEMBL14701105 0.85 MAPT (0.78) KMT2AMEN1RAD52BACE1DNM1
SCHEMBL14889275 0.84 BACE1 (1.00) KMT2AMEN1RAD52BACE1DNM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 183 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180318255-A1 Pro-Neurogenic Compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2018-11-08 US claimed
EP-2385829-B1 PRO-NEUROGENIC COMPOUNDS UNIV TEXAS (US) 2018-08-01 EP claimed
US-20170157092-A1 Anti-depression Compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2017-06-08 US claimed
US-9616048-B2 Anti-depression compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-04-11 US claimed
US-20160362372-A1 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2016-12-15 US claimed
US-20160206596-A1 Anti-depression Compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2016-07-21 US claimed
US-20160206594-A1 Pro-Neurogenic Compounds NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-07-21 US claimed
US-9162980-B2 Anti-depression compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-10-20 US claimed
US-20150290195-A1 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2015-10-15 US claimed
EP-2925129-A1 PRO-NEUROGENIC COMPOUNDS Board of Regents of the University of Texas System (US) 2015-10-07 EP claimed
EP-2590647-A2 PRO-NEUROGENIC COMPOUNDS Board of Regents of the University of Texas System (US) 2013-05-15 EP claimed
US-20130040977-A1 Pro-Neurogenic Compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2013-02-14 US claimed
US-8362277-B2 Pro-neurogenic compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-01-29 US claimed
US-20120022096-A1 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-01-26 US claimed
WO-2012006419-A2 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-01-12 WO claimed
EP-2385829-A1 PRO-NEUROGENIC COMPOUNDS Board of Regents of the University of Texas System (US) 2011-11-16 EP claimed
US-8039041-B2 Electroluminescent devices with electrode protection CAMBRIDGE DISPLAY TECHNOLOGY, LTD. (GB) 2011-10-18 US claimed
US-20110015217-A1 Pro-Neurogenic Compounds BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2011-01-20 US claimed
US-20110003836-A1 Pro-Neurogenic Compounds BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2011-01-06 US claimed
WO-2010081115-A1 PRO-NEUROGENIC COMPOUNDS UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER (US) 2010-07-15 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120022096-A1 PRO-NEUROGENIC COMPOUNDS BDNF, GAP43, DCX KMT2A 3749/4885MEN1 3423/4885RAD52 3297/4885
US-20160206594-A1 Pro-Neurogenic Compounds DCX, GAP43, BDNF KMT2A 2693/4885MEN1 3192/4885RAD52 4273/4885
US-20180318255-A1 Pro-Neurogenic Compounds BDNF, GAP43, DCX KMT2A 3749/4885MEN1 3423/4885RAD52 3297/4885
US-20110015217-A1 Pro-Neurogenic Compounds DCX, GAP43, BDNF KMT2A 2693/4885MEN1 3192/4885RAD52 4273/4885
US-20150290195-A1 PRO-NEUROGENIC COMPOUNDS DCX, GAP43, BDNF KMT2A 2693/4885MEN1 3192/4885RAD52 4273/4885
US-20130040977-A1 Pro-Neurogenic Compounds BDNF, GAP43, DCX KMT2A 3749/4885MEN1 3423/4885RAD52 3297/4885
US-20110003836-A1 Pro-Neurogenic Compounds DCX, GAP43, BDNF KMT2A 2838/4885MEN1 3234/4885RAD52 4298/4885
US-20160362372-A1 PRO-NEUROGENIC COMPOUNDS DCX, GAP43, BDNF KMT2A 2693/4885MEN1 3192/4885RAD52 4273/4885
US-20160206596-A1 Anti-depression Compounds BDNF, DCX, GAP43 KMT2A 3598/4885MEN1 4295/4885RAD52 2718/4885
US-20170157092-A1 Anti-depression Compounds BDNF, DCX, GAP43 KMT2A 3598/4885MEN1 4295/4885RAD52 2718/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.