SCHEMBL4119030

SCHEMBL4119030

COc1cc2c(-c3ccc(Br)cc3F)nc(N)nc2cc1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.47
EGFR P00533 3/20 0.45
ELANE P08246 1/20 0.44
CTSV O60911 1/20 0.42
CTSL P07711 1/20 0.42
ADORA2A P29274 1/20 0.42
KDM1A O60341 2/20 0.42
PDPK1 O15530 1/20 0.42
NSD2 O96028 1/20 0.42
RET P07949 1/20 0.41
KIF5B P33176 1/20 0.41
KDR P35968 1/20 0.41
TLR9 Q9NR96 2/20 0.41
TLR7 Q9NYK1 2/20 0.41
IRAK1 P51617 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
ATM Q13315 1/20 0.41
EHMT2 Q96KQ7 1/20 0.41
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4108476 0.79 EGFR (0.44) KITEGFRADORA2ARETKIF5B
SCHEMBL7791033 0.78 ADORA2A (0.61) KITEGFRADORA2ANSD2ATM
SCHEMBL13975080 0.77 ELANE (0.54) EGFRELANEKDM1APDPK1NSD2
SCHEMBL15502326 0.76 ELANE (0.53) EGFRELANEKDM1APDPK1NSD2
SCHEMBL7145589 0.76 TRPA1 (0.45) EGFRELANECTSVCTSLKDM1A
SCHEMBL4421590 0.74 TRPA1 (0.61) EGFRKDM1ARETKIF5BKDR
SCHEMBL21408242 0.73 MET (0.58) EGFRKDR
SCHEMBL30216641 0.73 MET (0.58) EGFRKDR
SCHEMBL7790971 0.73 ADORA2A (0.57) EGFRADORA2APDPK1ATM
SCHEMBL159652 0.73 KDR (0.80) KITEGFRRETKIF5BKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2613153-A2 Process for the identification of novel enzyme interacting compounds Cellzome GmbH (DE) 2013-07-10 EP disclosed
EP-2613154-A2 Process for the identification of novel enzyme interacting compounds Cellzome GmbH (DE) 2013-07-10 EP disclosed
EP-1891446-B1 PROCESS FOR THE IDENTIFICATION OF NOVEL ENZYME INTERACTING COMPOUNDS CELLZOME GMBH (DE) 2013-04-10 EP disclosed
US-20090238808-A1 Process for the identification of novel enzyme interacting compounds CELLZOME GMBH (DE) 2009-09-24 US disclosed
EP-1891446-A1 PROCESS FOR THE IDENTIFICATION OF NOVEL ENZYME INTERACTING COMPOUNDS CELLZOME AG (DE) 2008-02-27 EP disclosed
WO-2006134056-A1 PROCESS FOR THE IDENTIFICATION OF NOVEL ENZYME INTERACTING COMPOUNDS CELLZOME AG (DE) 2006-12-21 WO disclosed