Cerulenin

Cerulenin

SCHEMBL41207

C/C=C/C/C=C/CCC(=O)[C@H]1O[C@H]1C(N)=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 1.00
F13A1 P00488 4/20 1.00
MAPT P10636 3/20 1.00
PTGS1 P23219 2/20 1.00
THRB P10828 1/20 1.00
FASN P49327 1/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
CNR1 P21554 6/20 0.37
CYP19A1 P11511 2/20 0.36
RXRA P19793 2/20 0.36
PPARG P37231 2/20 0.36
OXER1 Q8TDS5 2/20 0.36
FFAR1 O14842 1/20 0.36
KDM4E B2RXH2 2/20 0.36
SOAT1 P35610 1/20 0.36
CNR2 P34972 4/20 0.33
TGM2 P21980 3/20 0.31
F7 P08709 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
F3 P13726 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cerulenin SCHEMBL20528755 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL3183350 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL8678332 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL4450603 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL28576416 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL10387308 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL8716153 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
SCHEMBL12902003 0.85 ALDH1A1 (0.74) ALDH1A1F13A1MAPTPTGS1THRB
SCHEMBL17874340 0.85 ALDH1A1 (0.74) ALDH1A1F13A1MAPTPTGS1THRB
SCHEMBL9453468 0.81 ALDH1A1 (0.68) ALDH1A1F13A1MAPTPTGS1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5920 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250297321-A1 METHOD FOR DETECTING METABOLIC REPROGRAMING OF CANCER TOWARDS FATTY ACIDS METABOLISM INST NAT SANTE RECH MED (FR) 2025-09-25 US claimed
US-20250263758-A1 A CELL-FREE BIO-MANUFACTURING PLATFORM FOR PRODUCTION OF FATTY ACIDS AND CANNABINOIDS UNITED STATES DEPARTMENT OF ENERGY 2025-08-21 US claimed
WO-2025151075-A1 METHODS OF TREATING CANCER AND COMBINATIONS THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2025-07-17 WO claimed
US-20250228841-A1 COMPOSITIONS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES APTORUM THERAPEUTICS LTD (HK) 2025-07-17 US claimed
WO-2025124485-A1 SCHIZOCHYTRIUM ALGAE STRAIN RICH IN N-3 FATTY ACID AND SCREENING AND CULTURE METHOD THEREFOR 厦门汇盛生物有限公司 2025-06-19 WO claimed
US-20250177367-A1 COMBINATION THERAPIES FOR MODULATION OF LIPID PRODUCTION OHIO STATE INNOVATION FOUNDATION 2025-06-05 US claimed
CN-119881339-A Serum metabonomics-based long-life biomarker and application thereof 广东医科大学 2025-04-25 CN claimed
WO-2025071221-A1 WICKERHAMOMYCES SP. MICROORGANISM HAVING HIGH PRODUCTIVITY OF PHYTOSPHINGOSINE DERIVATIVE 주식회사 케이씨아이 2025-04-03 WO claimed
CN-119677539-A Combination therapy for modulating lipid production 俄亥俄州创新基金会 2025-03-21 CN claimed
EP-4489865-A2 COMBINATION THERAPIES FOR MODULATION OF LIPID PRODUCTION Ohio State Innovation Foundation (US) 2025-01-15 EP claimed
WO-1995019706-A1 INHIBITORS OF FATTY ACID SYNTHESIS AS ANTIMICROBIAL AGENTS THE JOHNS HOPKINS UNIVERSITY (US) 1995-07-27 WO claimed
WO-1995019765-A1 CERTAIN CERULENIN-GERANYL AND DODECANOIC ACID DERIVATIVES CHEKTEC CORPORATION (US) 1995-07-27 WO claimed
EP-0585390-A4 STEALTH VIRUS DETECTION IN THE CHRONIC FATIGUE SYNDROME. MARTIN WILLIAM JOHN (US) 1995-05-31 EP claimed
EP-0651636-A1 CHEMOTHERAPY FOR CANCER THE JOHNS HOPKINS UNIVERSITY (US) 1995-05-10 EP claimed
EP-0585390-A1 STEALTH VIRUS DETECTION IN THE CHRONIC FATIGUE SYNDROME MARTIN, William John (US) 1994-03-09 EP claimed
WO-1994002108-A1 CHEMOTHERAPY FOR CANCER THE JOHNS HOPKINS UNIVERSITY (US) 1994-02-03 WO claimed
WO-1992020787-A1 STEALTH VIRUS DETECTION IN THE CHRONIC FATIGUE SYNDROME MARTIN WILLIAM JOHN (US) 1992-11-26 WO claimed
EP-0121408-B1 IMPROVEMENTS IN OR RELATING TO MACROLIDE ANTIBIOTICS Omura, Satoshi (JP) 1989-03-01 EP claimed
EP-0121408-A2 Improvements in or relating to macrolide antibiotics Omura, Satoshi (JP) 1984-10-10 EP claimed
EP-0074244-A1 Process for producing spiramycin I KYOWA HAKKO KOGYO CO., LTD. (JP) 1983-03-16 EP claimed