Cerulenin

Cerulenin

SCHEMBL8716153

CC=CCC=CCCC(=O)[C@@H]1OC1C(N)=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 1.00
F13A1 P00488 4/20 1.00
MAPT P10636 3/20 1.00
PTGS1 P23219 2/20 1.00
THRB P10828 1/20 1.00
FASN P49327 1/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
CNR1 P21554 6/20 0.37
CYP19A1 P11511 2/20 0.36
RXRA P19793 2/20 0.36
PPARG P37231 2/20 0.36
OXER1 Q8TDS5 2/20 0.36
FFAR1 O14842 1/20 0.36
KDM4E B2RXH2 2/20 0.36
SOAT1 P35610 1/20 0.36
CNR2 P34972 4/20 0.33
TGM2 P21980 3/20 0.31
F7 P08709 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
F3 P13726 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cerulenin SCHEMBL20528755 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL3183350 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL8678332 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL4450603 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL41207 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL28576416 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
Cerulenin SCHEMBL10387308 1.00 ALDH1A1 (1.00) ALDH1A1F13A1MAPTPTGS1THRB
SCHEMBL12902003 0.85 ALDH1A1 (0.74) ALDH1A1F13A1MAPTPTGS1THRB
SCHEMBL17874340 0.85 ALDH1A1 (0.74) ALDH1A1F13A1MAPTPTGS1THRB
SCHEMBL9453468 0.81 ALDH1A1 (0.68) ALDH1A1F13A1MAPTPTGS1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5759837-A ANTITUMOR AGENTS AND ANTICARCINOGENIC AGENTS JOHN HOPKINS UNIVERSITY (US) 1998-06-02 US disclosed
US-5614551-A Inhibitors of fatty acid synthesis as antimicrobial agents THE JOHNS HOPKINS UNIVERSITY (US) 1997-03-25 US disclosed
US-5539132-A Cerulenin compounds for fatty acid synthesis inhibition JOHNS HOPKINS UNIVERSITY (US) 1996-07-23 US disclosed
WO-1995019765-A1 CERTAIN CERULENIN-GERANYL AND DODECANOIC ACID DERIVATIVES CHEKTEC CORPORATION (US) 1995-07-27 WO disclosed
EP-0651636-A1 CHEMOTHERAPY FOR CANCER THE JOHNS HOPKINS UNIVERSITY (US) 1995-05-10 EP disclosed
WO-1994002108-A1 CHEMOTHERAPY FOR CANCER THE JOHNS HOPKINS UNIVERSITY (US) 1994-02-03 WO disclosed