SCHEMBL4122903

SCHEMBL4122903

Cc1ccc(NC(=O)Nc2ccccc2)cc1F

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.71
RAB9A P51151 6/20 0.71
KMT2A Q03164 6/20 0.66
MAPT P10636 4/20 0.66
MEN1 O00255 3/20 0.66
LMNA P02545 3/20 0.66
HTT P42858 2/20 0.66
STING1 Q86WV6 1/20 0.61
SMN1; SMN2 Q16637 4/20 0.60
MAPK1 P28482 1/20 0.60
FPR2 P25090 4/20 0.60
KCNJ6 P48051 1/20 0.57
KCNJ5 P48544 1/20 0.57
KCNJ3 P48549 1/20 0.57
TP53 P04637 1/20 0.57
EPHX1 P07099 1/20 0.57
TSHR P16473 1/20 0.57
EPHX2 P34913 1/20 0.57
CDK9 P50750 1/20 0.57
CLK4 Q9HAZ1 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4118553 0.91 NPC1 (0.69) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL4112443 0.88 NPC1 (0.71) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL4112362 0.88 NPC1 (0.67) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL4112024 0.87 NPC1 (0.63) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL4115751 0.87 NPC1 (0.67) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL4112951 0.87 NPC1 (0.61) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL4117300 0.86 NPC1 (0.67) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL4105335 0.86 NPC1 (0.64) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL4115616 0.86 NPC1 (0.65) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL4548132 0.85 IDH1 (0.64) NPC1RAB9AKMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4228630-B1 NLRP3 ACTIVATORS FOR USE IN THE TREATMENT OF INFECTIOUS DISEASES OR CANCER BY ACTIVATING NLRP3 INFLAMMASOME UNIV FREIBURG ALBERT LUDWIGS (DE) 2025-03-05 EP claimed
US-20240277658-A1 NLRP3 ACTIVATORS FOR USE IN THE TREATMENT OF INFECTIOUS DISEASES OR CANCER BY ACTIVATING NLRP3 INFLAMMASOME ALBERT-LUDWIGS-UNIVERSITÄT FREIBURG (DE) 2024-08-22 US claimed
EP-4228630-B1 NLRP3 ACTIVATORS FOR USE IN THE TREATMENT OF INFECTIOUS DISEASES OR CANCER BY ACTIVATING NLRP3 INFLAMMASOME UNIV FREIBURG ALBERT LUDWIGS (DE) 2025-03-05 EP disclosed
US-20240277658-A1 NLRP3 ACTIVATORS FOR USE IN THE TREATMENT OF INFECTIOUS DISEASES OR CANCER BY ACTIVATING NLRP3 INFLAMMASOME ALBERT-LUDWIGS-UNIVERSITÄT FREIBURG (DE) 2024-08-22 US disclosed
US-20090239841-A1 Diaryl Ureas as CB1 Antagonists NEUROGEN CORPORATION 2009-09-24 US disclosed
US-20090239841-A1 Diaryl Ureas as CB1 Antagonists NEUROGEN CORPORATION 2009-09-24 US disclosed
US-20090239841-A1 Diaryl Ureas as CB1 Antagonists NEUROGEN CORPORATION 2009-09-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090239841-A1 Diaryl Ureas as CB1 Antagonists CNR1, CNR2, OPRL1 NPC1 927/4885RAB9A 815/4885KMT2A 2807/4885
US-20240277658-A1 NLRP3 ACTIVATORS FOR USE IN THE TREATMENT OF INFECTIOUS DISEASES OR CANCER BY ACTIVATING NLRP3 INFLAMMASOME NLRP3, PYCARD, NLRP1 NPC1 146/4885RAB9A 2409/4885KMT2A 4020/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.