SCHEMBL4123024

SCHEMBL4123024

Cn1nc(C(C)(C)C)c2nc(N(CCCN3CCOCC3)CC3CCCCC3)[nH]c(=O)c21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.36
KDM4E B2RXH2 7/20 0.36
HPGD P15428 2/20 0.36
USP2 O75604 2/20 0.36
HSD17B10 Q99714 5/20 0.35
NPSR1 Q6W5P4 5/20 0.35
TSHR P16473 4/20 0.35
GAA P10253 2/20 0.35
ALOX15 P16050 2/20 0.34
TP53 P04637 1/20 0.34
CASP1 P29466 2/20 0.33
CASP7 P55210 2/20 0.33
PDE9A O76083 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.32
MAPT P10636 2/20 0.32
PKM P14618 2/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8034133 0.90 KDM4E (0.36) ALDH1A1KDM4EHPGDUSP2HSD17B10
SCHEMBL8042659 0.88 KDM4E (0.37) ALDH1A1KDM4EUSP2NPSR1TSHR
SCHEMBL8033607 0.87 KDM4E (0.36) ALDH1A1KDM4ENPSR1SMN1; SMN2MAPT
SCHEMBL4134627 0.86 MAPT (0.34) ALDH1A1KDM4EHPGDUSP2HSD17B10
SCHEMBL4131082 0.85 MAPT (0.34) ALDH1A1KDM4EHSD17B10NPSR1TSHR
SCHEMBL4132580 0.85 KDM4E (0.35) ALDH1A1KDM4ENPSR1SMN1; SMN2MAPT
SCHEMBL8045132 0.84 KDM4E (0.41) ALDH1A1KDM4ENPSR1SMN1; SMN2MAPT
SCHEMBL4139405 0.83 KDM4E (0.34) ALDH1A1KDM4ENPSR1SMN1; SMN2MAPT
SCHEMBL8049123 0.82 KDM4E (0.37) ALDH1A1KDM4ENPSR1SMN1; SMN2MAPT
SCHEMBL8043252 0.81 KDM4E (0.36) ALDH1A1KDM4ENPSR1PDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071707-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed