SCHEMBL413617

SCHEMBL413617

COCCNC(=O)c1ccc2nc(-c3cccc(C)n3)c(-c3ccnc(N)n3)n2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 4/20 0.50
AKT1 P31749 2/20 0.47
AKT2 P31751 2/20 0.47
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GLA P06280 2/20 0.43
HPGD P15428 2/20 0.43
CASP1 P29466 2/20 0.43
CASP7 P55210 2/20 0.43
HSD17B10 Q99714 2/20 0.43
TP53 P04637 1/20 0.43
GAA P10253 1/20 0.43
MAP3K14 Q99558 2/20 0.42
TRIM33 Q9UPN9 3/20 0.42
PIK3CD O00329 1/20 0.41
PIK3R1 P27986 1/20 0.41
IGF1R P08069 1/20 0.40
JAK2 O60674 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL409368 0.92 TGFBR1 (0.42) TGFBR1AKT1AKT2KDM4EALDH1A1
SCHEMBL409977 0.90 MAP3K14 (0.45) TGFBR1AKT1AKT2KDM4EHSD17B10
SCHEMBL407985 0.89 TGFBR1 (0.46) TGFBR1TP53MAP3K14PIK3CDPIK3R1
SCHEMBL412682 0.89 MAP3K14 (0.46) TGFBR1MAP3K14PIK3CDPIK3R1IGF1R
SCHEMBL27615221 0.88 MAP3K14 (0.41) TGFBR1AKT1AKT2KDM4EALDH1A1
SCHEMBL411998 0.87 MAP3K14 (0.47) TGFBR1AKT1AKT2MAP3K14PIK3CD
SCHEMBL412151 0.87 MAP3K14 (0.47) TGFBR1AKT1AKT2MAP3K14TRIM33
SCHEMBL412286 0.86 NPC1 (0.43) TGFBR1KDM4EALDH1A1HPGDTP53
SCHEMBL412220 0.85 TGFBR1 (0.43) TGFBR1KDM4ETP53MAP3K14PIK3CD
SCHEMBL413826 0.84 AKT1 (0.46) TGFBR1AKT1AKT2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120021519-A1 EFFICIENT INDUCTION OF PLURIPOTENT STEM CELLS USING SMALL MOLECULE COMPOUNDS PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-26 US disclosed