SCHEMBL4140165

SCHEMBL4140165

COc1ccc(C(=O)c2c(C)[nH]c3ccncc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.56
PTGS2 P35354 1/20 0.56
ACHE P22303 2/20 0.55
TUBB1 Q9H4B7 1/20 0.48
PIKFYVE Q9Y2I7 1/20 0.46
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
RAB9A P51151 2/20 0.44
CHUK O15111 2/20 0.44
PTPN5 P54829 1/20 0.44
ALDH1A1 P00352 1/20 0.43
JAK2 O60674 1/20 0.43
MAPT P10636 2/20 0.43
ICOSLG O75144 1/20 0.43
ICOS Q9Y6W8 1/20 0.43
KIF20A O95235 1/20 0.43
KDM4E B2RXH2 1/20 0.43
TLR3 O15455 1/20 0.43
NR3C1 P04150 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8531445 0.81 PTGS1 (0.64) PTGS1PTGS2TUBB1KMT2ARAB9A
SCHEMBL28524519 0.78 PTGS1 (0.62) PTGS1PTGS2TUBB1KMT2AMEN1
SCHEMBL30619664 0.77 NR4A2 (0.46) ACHERAB9AJAK2MAPT
SCHEMBL29587497 0.77 NR4A2 (0.46) ACHERAB9AJAK2MAPT
SCHEMBL8534628 0.76 PTGS1 (0.59) PTGS1PTGS2TUBB1KMT2AMEN1
SCHEMBL2974886 0.76 ALDH1A1 (0.61) PTGS1PTGS2TUBB1PIKFYVEKMT2A
SCHEMBL4135200 0.75 ACHE (0.56) PTGS2ACHEKMT2AMEN1RAB9A
SCHEMBL3236462 0.75 ACHE (0.47) ACHEKMT2AMEN1RAB9AALDH1A1
SCHEMBL25260242 0.74 ALDH1A1 (0.58) PTGS1PTGS2TUBB1KMT2AMEN1
SCHEMBL2972598 0.73 TUBB1 (0.70) PTGS1PTGS2TUBB1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009005672-A1 ANTIDIABETIC AZAINDOLES AND DIAZAINDOLES MERCK & CO., INC. (US) 2009-01-08 WO disclosed
WO-2009005672-A1 ANTIDIABETIC AZAINDOLES AND DIAZAINDOLES MERCK & CO., INC. (US) 2009-01-08 WO disclosed