SCHEMBL4141201

SCHEMBL4141201

COc1cc2c(Oc3ccc(C(N)=O)cc3)ccnc2cc1O

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 4/20 0.59
PDGFRA P16234 7/20 0.57
PDGFRB P09619 1/20 0.57
KDR P35968 7/20 0.56
MET P08581 4/20 0.56
AURKA O14965 2/20 0.56
TEK Q02763 2/20 0.56
AURKB Q96GD4 2/20 0.56
ABL1 P00519 1/20 0.56
LCK P06239 1/20 0.56
LYN P07948 1/20 0.56
KIT P10721 1/20 0.51
AXL P30530 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3794599 0.91 FGFR2 (0.69) FGFR2PDGFRAPDGFRBKDRMET
SCHEMBL4141203 0.85 FGFR2 (0.60) FGFR2PDGFRAPDGFRBKDR
SCHEMBL4575945 0.84 MET (0.52) FGFR2PDGFRAKDRMETKIT
SCHEMBL25678872 0.84 KDR (0.67) FGFR2PDGFRAPDGFRBKDRMET
SCHEMBL17489704 0.84 PDGFRA (0.65) FGFR2PDGFRAPDGFRBKDR
SCHEMBL17361401 0.83 MET (0.55) PDGFRAKDRMETKITAXL
SCHEMBL12499486 0.82 FGFR2 (0.56) FGFR2PDGFRAPDGFRBKDRMET
SCHEMBL14967576 0.82 MET (0.60) FGFR2PDGFRAPDGFRBKDRMET
SCHEMBL4154997 0.81 PDGFRA (0.59) FGFR2PDGFRAPDGFRBKDRMET
SCHEMBL28428907 0.81 PDGFRA (0.55) FGFR2PDGFRAPDGFRBKDRMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090131461-A1 Quinoline and quinoxaline derivatives as inhibitors of kinase enzymatic activity CHROMA THERAPEUTICS LTD. (GB) 2009-05-21 US disclosed
EP-1877383-A1 QUINOLINE AND QUINOXALINE DERIVATIVES AS INHIBITORS OF KINASE ENZYMATIC ACTIVITY Chroma Therapeutics Limited (GB) 2008-01-16 EP disclosed
WO-2006117552-A1 QUINOLINE AND QUINOXALINE DERIVATIVES AS INHIBITORS OF KINASE ENZYMATIC ACTIVITY CHROMA THERAPEUTICS LTD (GB) 2006-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090131461-A1 Quinoline and quinoxaline derivatives as inhibitors of kinase enzymatic activity CDK1, AURKC, CSNK1G3 FGFR2 3819/4885PDGFRA 3858/4885PDGFRB 3487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.