SCHEMBL4145291

SCHEMBL4145291

COC(=O)c1ccc2c(c1)N=Cc1c(Cl)cccc1S2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.44
TRPA1 O75762 5/20 0.44
TP53 P04637 4/20 0.41
MAPT P10636 3/20 0.39
CNR1 P21554 2/20 0.39
CNR2 P34972 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PFKFB3 Q16875 1/20 0.38
PFKFB4 Q16877 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4146312 0.84 CNR1 (0.46) TP53MAPTCNR1CNR2KDM4E
SCHEMBL4146318 0.84 CNR1 (0.35) POLBTP53MAPTCNR1CNR2
SCHEMBL4147214 0.84 PARP1 (0.40) TP53MAPTCNR1CNR2
SCHEMBL4670768 0.74 PLEC (0.53) POLBTP53MAPTCNR1CNR2
SCHEMBL11397180 0.73 TRPA1 (0.63) TRPA1TP53MAPTALDH1A1KDM4E
SCHEMBL1726796 0.72 TRPA1 (0.56) TRPA1
SCHEMBL4668625 0.71 SIRT2 (0.39) POLBTP53MAPTCNR1CNR2
SCHEMBL9511152 0.71 KDM4E (0.52) POLBTP53MAPTALDH1A1KDM4E
SCHEMBL4808618 0.70 CHEK2 (0.43)
SCHEMBL11387022 0.69 TP53 (0.43) POLBTRPA1TP53MAPTCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009075691-A1 CB-1 MODULATING COMPOUNDS AND THEIR USE ACADIA PHARMACEUTICALS INC. (US) 2009-06-18 WO disclosed
WO-2008118141-A2 USE OF CANNABINOID MODULATING COMPOUNDS IN COMBINATION WITH OTHER THERAPEUTIC COMPOUNDS FOR ADJUNCTIVE THERAPY ACADIA PHARMACEUTICALS INC. (US) 2008-10-02 WO disclosed
EP-1937614-A1 IRON CATALYZED CROSS-COUPLING REACTIONS OF IMIDOYL DERIVATIVES Arcadia Pharmaceuticals Inc. (US) 2008-07-02 EP disclosed
WO-2007047776-A1 IRON CATALYZED CROSS-COUPLING REACTIONS OF IMIDOYL DERIVATIVES ACADIA PHARMACEUTICALS INC. (US) 2007-04-26 WO disclosed