SCHEMBL414592

SCHEMBL414592

CCOCCCNC(=O)c1ccc2c(-c3c(-c4cccc(C)n4)nn4ccccc34)ccnc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 10/20 0.47
KMT2A Q03164 3/20 0.45
MAPK14 Q16539 2/20 0.43
THRB P10828 1/20 0.43
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 2/20 0.41
KDR P35968 3/20 0.41
NPC1 O15118 1/20 0.41
GAK O14976 1/20 0.41
RIPK2 O43353 1/20 0.41
MAP4K4 O95819 1/20 0.41
ACVR1B P36896 1/20 0.41
TGFBR2 P37173 1/20 0.41
CSNK1A1 P48729 1/20 0.41
CSNK1D P48730 1/20 0.41
CSNK1E P49674 1/20 0.41
TGFB2 P61812 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL413710 0.90 TGFBR1 (0.49) TGFBR1KMT2AMAPK14THRBALDH1A1
SCHEMBL412491 0.89 TGFBR1 (0.57) TGFBR1MAPK14THRBALDH1A1HPGD
SCHEMBL414681 0.89 TGFBR1 (0.51) TGFBR1KMT2AMAPK14THRBALDH1A1
SCHEMBL5238981 0.89 TGFBR1 (0.47) TGFBR1MAPK14THRBKDRGAK
SCHEMBL412319 0.87 TGFBR1 (0.61) TGFBR1MAPK14THRBKDRGAK
SCHEMBL414211 0.86 TGFBR1 (0.53) TGFBR1KMT2AMAPK14THRBALDH1A1
SCHEMBL412295 0.86 NAMPT (0.50) ALDH1A1NAMPT
SCHEMBL412977 0.86 TGFBR1 (0.51) TGFBR1MAPK14THRBKDRGAK
SCHEMBL413597 0.86 TGFBR1 (0.48) TGFBR1MAPK14THRBKDRGAK
SCHEMBL409683 0.85 TGFBR1 (0.48) TGFBR1KMT2AMAPK14SMN1; SMN2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120021519-A1 EFFICIENT INDUCTION OF PLURIPOTENT STEM CELLS USING SMALL MOLECULE COMPOUNDS PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-26 US disclosed