Glutarate

Glutarate

SCHEMBL4148651

N=C(N)N.N=C(N)N.O=C(O)CCCC(=O)O

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2

The experimentally established mechanism targets of Glutarate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A6 Q4U2R8 1/20 0.69
LMNA P02545 5/20 0.59
TSHR P16473 3/20 0.56
NFKB1 P19838 2/20 0.56
PMP22 Q01453 1/20 0.56
THRB P10828 2/20 0.55
BLM P54132 2/20 0.55
KMT2A Q03164 2/20 0.55
NPSR1 Q6W5P4 2/20 0.55
GABRR3 A8MPY1 1/20 0.55
GABRP O00591 1/20 0.55
GABRD O14764 1/20 0.55
HDAC3 O15379 1/20 0.55
GABBR2 O75899 1/20 0.55
CYP1A2 P05177 1/20 0.55
GABRA1 P14867 1/20 0.55
GABRB1 P18505 1/20 0.55
GABRG2 P18507 1/20 0.55
GABRR1 P24046 1/20 0.55
GABRB3 P28472 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Adipic Acid SCHEMBL1071331 0.94 LMNA (0.69) SLC22A6LMNATSHRNFKB1PMP22
Adipic Acid SCHEMBL28047756 0.91 LMNA (0.65) SLC22A6LMNATSHRNFKB1PMP22
SCHEMBL1736025 0.88
Succinic Acid SCHEMBL1071158 0.87 LMNA (0.64) SLC22A6LMNATSHRNFKB1PMP22
Glutarate SCHEMBL2875088 0.87 SLC22A6 (0.79) SLC22A6LMNATSHRNFKB1PMP22
SCHEMBL436313 0.84
Valeric Acid SCHEMBL31741355 0.84 AKR1B1 (0.64) SLC22A6LMNATSHRBLMKMT2A
Glutarate SCHEMBL30862146 0.84 SLC22A6 (0.55) SLC22A6LMNATSHRNFKB1PMP22
Gamma-Aminobutyric Acid SCHEMBL28266648 0.84 LMNA (0.75) SLC22A6LMNATSHRNFKB1PMP22
Glutarate SCHEMBL3911885 0.83 SLC22A6 (0.85) SLC22A6LMNATSHRNFKB1PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090242236-A1 METHOD OF FORMING CONDUCTIVE TRACKS EASTMAN KODAK COMPANY 2009-10-01 US disclosed
US-20090142559-A1 METHOD OF FORMING CONDUCTIVE TRACKS FOR FLEXIBLE ELECTRONIC CIRCUITS EASTMAN KODAK COMPANY 2009-06-04 US disclosed
US-20080290084-A1 Method of Forming a Flexible Heating Element CITICORP NORTH AMERICA, INC., AS AGENT 2008-11-27 US disclosed
US-7449286-B2 Method of forming conductive tracks EASTMAN KODAK COMPANY (US) 2008-11-11 US disclosed
EP-1932057-A2 METHOD OF FORMING CONDUCTIVE TRACKS EASTMAN KODAK COMPANY (US) 2008-06-18 EP disclosed
EP-1932402-A1 METHOD OF FORMING CONDUCTIVE TRACKS FOR FLEXIBLE ELECTRONIC CIRCUITS EASTMAN KODAK COMPANY (US) 2008-06-18 EP disclosed
EP-1932392-A2 METHOD OF FORMING A FLEXIBLE HEATING ELEMENT EASTMAN KODAK COMPANY (US) 2008-06-18 EP disclosed
WO-2007031710-A2 METHOD OF FORMING A FLEXIBLE HEATING ELEMENT EASTMAN KODAK COMPANY (US) 2007-03-22 WO disclosed
WO-2007031711-A1 METHOD OF FORMING CONDUCTIVE TRACKS FOR FLEXIBLE ELECTRONIC CIRCUITS EASTMAN KODAK COMPANY (US) 2007-03-22 WO disclosed
WO-2007031712-A2 METHOD OF FORMING CONDUCTIVE TRACKS EASTMAN KODAK COMPANY (US) 2007-03-22 WO disclosed
US-6492076-B1 UNDERGOES CHANGE IN ELECTROMAGNETIC ABSORPTION WHEN HEATED; ANTIHALATION OR FILTER LAYERS CONTAINING ZWITTERIONIC 1-AMINOPYRIDINIUM DYE EASTMAN KODAK COMPANY 2002-12-10 US disclosed
US-6455210-B1 SUPPORT, PHOTOTHERMOGRAPHIC IMAGE- RECEIVING LAYERS, AND ANTIHALATION LAYER OR FILTER LAYERS OF A DYE AND A HEXAARYLBIIMIDAZOLE IN A DISPERSION OF A HYDROPHILIC POLYMER EASTMAN KODAK COMPANY 2002-09-24 US disclosed
US-6451516-B1 AMINOPYRIDINIUM DYE WITH METHIN LINKAGE TERMINATED BY A HETEROCVYCLIC NUCLEUS AS FOUND IN CYANINE DYES EASTMAN KODAK COMPANY 2002-09-17 US disclosed
US-20020106590-A1 AQUEOUS THERMALLY BEACHABLE COMPOSITION USEFUL IN A PHOTOTHERMOGRAPHIC ELEMENT CARESTREAM HEALTH, INC. 2002-08-08 US disclosed
EP-1217431-A2 An aqueous thermally bleachable composition useful in a photothermographic element EASTMAN KODAK COMPANY (US) 2002-06-26 EP disclosed
US-4201590-A Heat sensitive reactive products of hexaarylbiimidazole and antihalation dyes EASTMAN KODAK COMPANY (US) 1980-05-06 US disclosed
US-4196002-A HEXAARYLBISMIIDAZOLE, COLORLESS EASTMAN KODAK COMPANY (US) 1980-04-01 US disclosed
US-4088496-A SILVER SALT, DEVELOPER, BINDER AND AN ACTIVATOR, THE ACID PORTION OF WHICH IS 2-CARBOXYCARBOXAMIDE EASTMAN KODAK COMPANY (US) 1978-05-09 US disclosed
US-4060420-A PHOTOGRAPHY EASTMAN KODAK COMPANY (US) 1977-11-29 US disclosed
US-4012260-A THIAZOLINIUM COMPOUNDS EASTMAN KODAK COMPANY (US) 1977-03-15 US disclosed