Buspirone

Buspirone

SCHEMBL41495

Cl.O=C1CC2(CCCC2)CC(=O)N1CCCCN1CCN(c2ncccn2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HTR1A

The experimentally established mechanism targets of Buspirone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A known ✓ P08908 8/20 0.98
ALDH1A1 P00352 2/20 1.00
KDM4E B2RXH2 1/20 1.00
PMP22 Q01453 1/20 1.00
DRD2 P14416 2/20 0.98
HTR2A P28223 2/20 0.98
SLC22A2 O15244 1/20 0.98
ABCB11 O95342 1/20 0.98
CYP1A2 P05177 1/20 0.98
CYP3A4 P08684 1/20 0.98
CYP2D6 P10635 1/20 0.98
CYP2C9 P11712 1/20 0.98
ADRA2C P18825 1/20 0.98
CNR1 P21554 1/20 0.98
ADRA1D P25100 1/20 0.98
HTR2C P28335 1/20 0.98
HTR7 P34969 1/20 0.98
ADRA1A P35348 1/20 0.98
HRH1 P35367 1/20 0.98
ADRA1B P35368 1/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Buspirone SCHEMBL10441318 1.00 ALDH1A1 (1.00) ALDH1A1KDM4EPMP22HTR1ADRD2
Hydrochloric Acid SCHEMBL11880141 0.99 ALDH1A1 (0.98) ALDH1A1KDM4EPMP22HTR1ADRD2
Hydrochloric Acid SCHEMBL11878911 0.99 ALDH1A1 (0.98) ALDH1A1KDM4EPMP22HTR1ADRD2
Buspirone SCHEMBL16398 0.99 HTR1A (1.00) ALDH1A1KDM4EPMP22HTR1ADRD2
Buspirone SCHEMBL17004050 0.99 HTR1A (1.00) ALDH1A1KDM4EPMP22HTR1ADRD2
Hydrochloric Acid SCHEMBL11877578 0.98 ALDH1A1 (0.95) ALDH1A1KDM4EPMP22HTR1ADRD2
SCHEMBL11875965 0.98 HTR1A (0.98) ALDH1A1KDM4EPMP22HTR1ADRD2
Buspirone SCHEMBL41496 0.98 HTR1A (0.98) ALDH1A1KDM4EPMP22HTR1ADRD2
SCHEMBL11875345 0.98 HTR1A (0.98) ALDH1A1KDM4EPMP22HTR1ADRD2
SCHEMBL11881209 0.96 HTR1A (0.95) ALDH1A1KDM4EPMP22HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2868 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-121578093-A Self-checking method of boost circuit, self-checking method of circuit and device thereof 上能电气股份有限公司 2026-02-27 CN claimed
CN-111342836-B Two-bus code sending driving circuit with protection control function 深圳市泰和安科技有限公司 2025-06-03 CN claimed
CN-119798224-A Preparation method of buspirone hydrochloride 山东京卫制药有限公司 2025-04-11 CN claimed
CN-119409681-A Preparation method of buspirone hydrochloride 北京华素制药股份有限公司 2025-02-11 CN claimed
CN-119198934-A Method and system for detecting residual solvent of buspirone hydrochloride solvent 武汉海特生物创新医药研究有限公司 2024-12-27 CN claimed
CN-119023833-A Method and system for detecting related substances of buspirone hydrochloride starting material 武汉海特生物创新医药研究有限公司 2024-11-26 CN claimed
CN-118845719-A Melatonin/buspirone hydrochloride oral instant film agent and preparation method thereof 沈阳药科大学 2024-10-29 CN claimed
CN-118702676-A Preparation method of buspirone hydrochloride crystal form II 济南大学 2024-09-27 CN claimed
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
CN-115065299-B Neutral point voltage balancing method applied to control of three-level permanent magnet synchronous motor 冶金自动化研究设计院有限公司 2024-08-16 CN claimed
EP-0276543-A2 Use of buspirone for the improvement of short term memory Bristol-Myers Squibb Company (US) 1988-08-03 EP claimed
EP-0276536-A2 Use of buspirone for the improvement of short term memory Bristol-Myers Squibb Company (US) 1988-08-03 EP claimed
US-4687772-A Method for improvement of short term memory BRISTOL-MYERS COMPANY (US) 1987-08-18 US claimed
WO-1987004621-A1 TREATMENT OF SEXUAL DYSFUNCTION WITH BUSPIRONE OTHMER EKKEHARD (US) 1987-08-13 WO claimed
EP-0220696-A2 Use of buspirone for preparing pharmaceutical compositions for alleviation of phobic anxiety Bristol-Myers Squibb Company (US) 1987-05-06 EP claimed
US-4640921-A GENERALIZED ANXIETY DISORDER BRISTOL-MYERS (US) 1987-02-03 US claimed
US-4634703-A Method for alleviation of panic disorders BRISTOL-MYERS COMPANY (US) 1987-01-06 US claimed
US-4438119-A BUSPIRONE OR SALTS THEREOF MEAD JOHNSON & COMPANY (US) 1984-03-20 US claimed
US-4182763-A PALLIATIVE TREATMENT OF NEUROSES MEAD JOHNSON & COMPANY (US) 1980-01-08 US claimed
US-3976776-A Tranquilizer process employing N-(heteroarcyclic)piperazinylalkylazaspiroalkanediones MEAD JOHNSON & COMPANY (US) 1976-08-24 US claimed