SCHEMBL4153552

SCHEMBL4153552

NS(=O)(=O)c1cccc(Nc2nccc(-c3nccs3)n2)c1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SYK P43405 9/20 0.67
CDK2 P24941 7/20 0.66
SRC P12931 2/20 0.66
ZAP70 P43403 2/20 0.66
CDK1 P06493 8/20 0.60
CCNT1 O60563 5/20 0.60
CCNB1 P14635 5/20 0.60
CDK9 P50750 5/20 0.60
CCNA2 P20248 4/20 0.60
CDK7 P50613 4/20 0.60
CCNH P51946 4/20 0.60
CCNA1 P78396 4/20 0.60
SLC2A1 P11166 1/20 0.59
MTOR P42345 4/20 0.57
SMG1 Q96Q15 4/20 0.57
IKBKB O14920 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13924492 0.86 SYK (0.68) SYKCDK2SRCZAP70CDK1
SCHEMBL13924445 0.81 SYK (0.75) SYKCDK2SRCZAP70
SCHEMBL7524252 0.80 CDK1 (0.69) SYKCDK2SRCCDK1CCNT1
SCHEMBL7464681 0.80 CDK1 (0.61) SYKCDK2CDK1CCNT1CCNB1
SCHEMBL13924480 0.80 SYK (0.69) SYKCDK2SRCZAP70CDK9
SCHEMBL13924456 0.80 SYK (0.73) SYKCDK2SRCZAP70
SCHEMBL13924470 0.80 SYK (0.73) SYKCDK2SRCZAP70
SCHEMBL13924459 0.80 SYK (0.73) SYKCDK2SRCZAP70
SCHEMBL13924432 0.80 SYK (1.00) SYKCDK2SRCZAP70CDK1
SCHEMBL13924468 0.80 SYK (0.73) SYKCDK2SRCZAP70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US claimed
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WNT1, CTNNB1, WNT3A SYK 3093/4885CDK2 116/4885SRC 1155/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.