Nitric Acid

Nitric Acid

SCHEMBL4154314

COc1cccc(NS(=O)(=O)c2cccc(NC(=N)N)c2)c1.O=[N+]([O-])O

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ERG11

The experimentally established mechanism targets of Nitric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.59
LMNA P02545 2/20 0.59
HDAC3 O15379 1/20 0.52
HDAC4 P56524 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC7 Q8WUI4 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC10 Q969S8 1/20 0.52
HDAC11 Q96DB2 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
HDAC9 Q9UKV0 1/20 0.52
HDAC5 Q9UQL6 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.51
PKM P14618 3/20 0.51
HPGD P15428 1/20 0.51
F2 P00734 1/20 0.51
TP53 P04637 1/20 0.50
CYP19A1 P11511 1/20 0.50
POLB P06746 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nitric Acid SCHEMBL1363033 0.87 PLAU (0.54) ALDH1A1LMNASMN1; SMN2PKMTP53
Nitric Acid SCHEMBL2075198 0.80 LMNA (0.48) ALDH1A1LMNASMN1; SMN2POLBMAPT
SCHEMBL1185724 0.78 SIGMAR1 (0.62) ALDH1A1LMNASMN1; SMN2PKMTP53
Methane SCHEMBL28113069 0.77 SIGMAR1 (0.60) ALDH1A1LMNASMN1; SMN2PKMTP53
Bicarbonate SCHEMBL8492631 0.76 NPC1 (0.61) ALDH1A1LMNASMN1; SMN2PKMTP53
Bicarbonate SCHEMBL27820322 0.76 NPC1 (0.61) ALDH1A1LMNASMN1; SMN2PKMTP53
SCHEMBL2240850 0.75 CYP19A1 (0.65) ALDH1A1LMNASMN1; SMN2PKMHPGD
Nitrous Acid SCHEMBL5998989 0.74 SIGMAR1 (0.58) ALDH1A1LMNASMN1; SMN2PKMHPGD
SCHEMBL7785609 0.74 LMNA (0.45) ALDH1A1LMNASMN1; SMN2PKMF2
SCHEMBL8711296 0.74 CYP19A1 (0.88) ALDH1A1LMNASMN1; SMN2PKMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090137572-A1 2-substituted-4-heteroaryl-pyrimidines useful for the treatment of proliferative disorders CYCLACEL LIMITED (GB) 2009-05-28 US disclosed
EP-1756098-A2 2-SUBSTITUTED-4-HETEROARYL-PYRIMIDINES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISORDERS Cyclacel Limited (GB) 2007-02-28 EP disclosed
WO-2005116025-A2 2-SUBSTITUTED-4-HETEROARYL-PYRIMIDINES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISORDERS CYCLACEL LIMITED (GB) 2005-12-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090137572-A1 2-substituted-4-heteroaryl-pyrimidines useful for the treatment of proliferative disorders CDK2, CDK4, CDK20 ALDH1A1 2743/4885LMNA 1768/4885HDAC3 3442/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.