SCHEMBL416660

SCHEMBL416660

Cc1nnc(-c2cccc(Cl)c2)[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.53
MGAM O43451 1/20 0.53
SI P14410 1/20 0.53
MGAM2 Q2M2H8 1/20 0.53
ALDH1A1 P00352 2/20 0.51
KDM4E B2RXH2 1/20 0.51
MPI P34949 1/20 0.51
GFER P55789 1/20 0.51
PIN1 Q13526 1/20 0.50
HRH1 P35367 1/20 0.50
IDO1 P14902 4/20 0.49
NPY5R Q15761 1/20 0.48
SCN2A Q99250 1/20 0.45
IKBKE Q14164 1/20 0.44
POLB P06746 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
TYMP P19971 1/20 0.43
NPBWR1 P48145 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
MAPK13 O15264 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL416478 0.81 NR1I3 (0.50) ALDH1A1PIN1IDO1NPY5RTYMP
SCHEMBL31429182 0.79 HRH1 (0.50) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL1077128 0.79 NPC1 (0.51) GAAALDH1A1KDM4EGFERPOLB
Water SCHEMBL17103297 0.77 NPC1 (0.50) GAAALDH1A1KDM4EGFERPOLB
SCHEMBL3825940 0.77 HRH1 (0.56) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL415765 0.77 MAPK1 (0.47) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL416435 0.77 POLB (0.60) GAAALDH1A1KDM4EPIN1NPY5R
SCHEMBL418276 0.76 HRH1 (0.49) ALDH1A1KDM4EHRH1NPY5RTYMP
SCHEMBL416539 0.76 CYP1A2 (0.52) PIN1NPY5RTYMPMAPK13RAF1
SCHEMBL12130385 0.75 GAA (0.47) GAAMGAMSIMGAM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2012-01-26 US claimed
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2009-11-26 US claimed
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2012-01-26 US disclosed
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2012-01-26 US disclosed
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2012-01-26 US disclosed
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2009-11-26 US disclosed
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2009-11-26 US disclosed
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2009-11-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION CDH1, EPCAM, ICAM1 GAA 4332/4885MGAM 3243/4885SI 1695/4885
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION CDH1, EPCAM, ICAM1 GAA 4332/4885MGAM 3243/4885SI 1695/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.